日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of a small molecule that inhibits Bcl-3-mediated cyclin D1 expression in melanoma cells

发现一种能抑制黑色素瘤细胞中Bcl-3介导的细胞周期蛋白D1表达的小分子

Saamarthy, Karunakar; Ahlqvist, Kristofer; Daams, Renée; Balagunaseelan, Navisraj; Rinaldo-Matthis, Agnes; Kazi, Julhash U; Sime, Wondossen; Massoumi, Ramin

Phosphorylation of Leukotriene C4 Synthase at Serine 36 Impairs Catalytic Activity

白三烯 C4 合酶第 36 位丝氨酸的磷酸化削弱催化活性

Shabbir Ahmad, A Jimmy Ytterberg, Madhuranayaki Thulasingam, Fredrik Tholander, Tomas Bergman, Roman Zubarev, Anders Wetterholm, Agnes Rinaldo-Matthis, Jesper Z Haeggström

Catalytic Conversion of Lipophilic Substrates by Phase constrained Enzymes in the Aqueous or in the Membrane Phase

水相或膜相中相约束酶对亲脂性底物的催化转化

Cebula, Marcus; Turan, Ilke Simsek; Sjödin, Birgitta; Thulasingam, Madhuranayaki; Brock, Joseph; Chmyrov, Volodymyr; Widengren, Jerker; Abe, Hiroshi; Mannervik, Bengt; Haeggström, Jesper Z; Rinaldo-Matthis, Agnes; Akkaya, Engin U; Morgenstern, Ralf

Structural and Functional Analysis of Calcium Ion Mediated Binding of 5-Lipoxygenase to Nanodiscs

钙离子介导的 5-脂氧合酶与纳米圆盘结合的结构和功能分析

Ramakrishnan B Kumar, Lin Zhu, Helena Idborg, Olof Rådmark, Per-Johan Jakobsson, Agnes Rinaldo-Matthis, Hans Hebert, Caroline Jegerschöld

A dynamic Asp-Arg interaction is essential for catalysis in microsomal prostaglandin E2 synthase

动态 Asp-Arg 相互作用对于微粒体前列腺素 E2 合酶的催化至关重要

Joseph S Brock, Mats Hamberg, Navisraj Balagunaseelan, Michael Goodman, Ralf Morgenstern, Emilia Strandback, Bengt Samuelsson, Agnes Rinaldo-Matthis, Jesper Z Haeggström

Binding of Pro-Gly-Pro at the active site of leukotriene A4 hydrolase/aminopeptidase and development of an epoxide hydrolase selective inhibitor

Pro-Gly-Pro 与白三烯 A4 水解酶/氨基肽酶活性位点的结合及环氧化物水解酶选择性抑制剂的开发

Alena Stsiapanava, Ulrika Olsson, Min Wan, Thea Kleinschmidt, Dorothea Rutishauser, Roman A Zubarev, Bengt Samuelsson, Agnes Rinaldo-Matthis, Jesper Z Haeggström

A picomolar transition state analogue inhibitor of MTAN as a specific antibiotic for Helicobacter pylori

一种皮摩尔级过渡态类似物抑制剂,可作为MTAN的特异性抗生素用于治疗幽门螺杆菌感染

Wang, Shanzhi; Haapalainen, Antti M; Yan, Funing; Du, Quan; Tyler, Peter C; Evans, Gary B; Rinaldo-Matthis, Agnes; Brown, Rosemary L; Norris, Gillian E; Almo, Steven C; Schramm, Vern L

Transition state analogs of 5'-methylthioadenosine nucleosidase disrupt quorum sensing

5'-甲基硫代腺苷核苷酶的过渡态类似物会破坏群体感应。

Gutierrez, Jemy A; Crowder, Tamara; Rinaldo-Matthis, Agnes; Ho, Meng-Chiao; Almo, Steven C; Schramm, Vern L