日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

VMY-1-103 is a novel CDK inhibitor that disrupts chromosome organization and delays metaphase progression in medulloblastoma cells

VMY-1-103 是一种新型 CDK 抑制剂,它能破坏髓母细胞瘤细胞的染色体结构并延缓中期进程。

Ringer, Lymor; Sirajuddin, Paul; Heckler, Mary; Ghosh, Anup; Suprynowicz, Frank; Yenugonda, Venkata M; Brown, Milton L; Toretsky, Jeffrey A; Uren, Aykut; Lee, YiChien; MacDonald, Tobey J; Rodriguez, Olga; Glazer, Robert I; Schlegel, Richard; Albanese, Chris

VMY-1-103, a dansylated analog of purvalanol B, induces caspase-3-dependent apoptosis in LNCaP prostate cancer cells.

VMY-1-103 是 purvalanol B 的丹酰化类似物,可诱导 LNCaP 前列腺癌细胞发生 caspase-3 依赖性凋亡

Ringer Lymor, Sirajuddin Paul, Yenugonda Venkata Mahidhar, Ghosh Anup, Divito Kyle, Trabosh Valerie, Patel Yesha, Brophy Amanda, Grindrod Scott, Lisanti Michael P, Rosenthal Dean, Brown Milton L, Avantaggiati Maria Laura, Rodriguez Olga, Albanese Chris