日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Second-Generation AURKA-Targeting PROTACs: Structural Optimization toward in Vivo Degradation in Neuroblastoma

第二代靶向AURKA的PROTAC:针对神经母细胞瘤体内降解的结构优化

Krols, Simon; Rishfi, Muhammad; Martens, Fien; Van Hauwermeiren, Anouk; Sanders, Ellen; De Sutter, Pieter-Jan; Vermeulen, An; De Wever, Kaat; Bekaert, Sarah-Lee; Dolman, M Emmy M; Tax, Gabor; Kamili, Alvin; Fletcher, Jamie I; Depestel, Lisa; De Wilde, Bram; Durinck, Kaat; Van Calenbergh, Serge

RRM2 enhances MYCN-driven neuroblastoma formation and acts as a synergistic target with CHK1 inhibition

RRM2 增强 MYCN 驱动的神经母细胞瘤形成,并与 CHK1 抑制一起充当协同靶点

Carolina Nunes, Lisa Depestel, Liselot Mus, Kaylee M Keller, Louis Delhaye, Amber Louwagie, Muhammad Rishfi, Alex Whale, Neesha Kara, Simon R Andrews, Filemon Dela Cruz, Daoqi You, Armaan Siddiquee, Camila Takeno Cologna, Sam De Craemer, Emmy Dolman, Christoph Bartenhagen, Fanny De Vloed, Ellen Sand

Whole transcriptome profiling of liquid biopsies from tumour xenografted mouse models enables specific monitoring of tumour-derived extracellular RNA

对肿瘤异种移植小鼠模型液体活检样本进行全转录组分析,可以特异性地监测肿瘤来源的细胞外RNA

Vanessa Vermeirssen ,Jill Deleu ,Annelien Morlion ,Celine Everaert ,Jilke De Wilde ,Jasper Anckaert ,Kaat Durinck ,Justine Nuytens ,Muhammad Rishfi ,Frank Speleman ,Hanne Van Droogenbroeck ,Kimberly Verniers ,Maria Francesca Baietti ,Maarten Albersen ,Eleonora Leucci ,Edward Post ,Myron G Best ,Tom Van Maerken ,Bram De Wilde ,Jo Vandesompele ,Anneleen Decock