日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Long-Term Latency of Highly Mutated Cells in Normal Mouse Skin Is Reversed by Exposure to Tumor Promoters and Chronic Tissue Damage

正常小鼠皮肤中高度突变细胞的长期潜伏状态可通过暴露于肿瘤促进剂和慢性组织损伤而逆转。

Li, Yun Rose; Kandyba, Eve; Halliwill, Kyle; Delrosario, Reyno; Tran, Quan; Bayani, Nora; Wu, Di; Mirzoeva, Olga K; Reeves, Melissa Quino; Islam, S M Ashiqul; Riva, Laura; Bergstrom, Erik N; Achanta, Kavya; DiGiovanni, John; Alexandrov, Ludmil B; Balmain, Allan

Global siRNA screen identifies human host factors critical for SARS-CoV-2 replication and late stages of infection.

全球 siRNA 筛选确定了对 SARS-CoV-2 复制和感染后期至关重要的人类宿主因子

Yin Xin, Pu Yuan, Yuan Shuofeng, Pache Lars, Churas Christopher, Weston Stuart, Riva Laura, Simons Lacy M, Cisneros William J, Clausen Thomas, Biddle Grace, Doss-Gollin Simon, Deming Meagan, De Jesus Paul D, Kim Ha Na, Fuentes Daniel, Whitelock John M, Esko Jeffrey D, Lord Megan S, Mena Ignacio, García-Sastre Adolfo, Hultquist Judd F, Frieman Matthew B, Ideker Trey, Pratt Dexter, Martin-Sancho Laura, Chanda Sumit K

Optimization of a micro-scale air-liquid-interface model of human proximal airway epithelium for moderate throughput drug screening for SARS-CoV-2

优化用于中等通量SARS-CoV-2药物筛选的人类近端气道上皮微尺度气液界面模型

Sen, Chandani; Rickabaugh, Tammy M; Jeyachandran, Arjit Vijey; Yuen, Constance; Ghannam, Maisam; Durra, Abdo; Aziz, Adam; Castillo, Kristen; Garcia, Gustavo Jr; Purkayastha, Arunima; Han, Brandon; Boulton, Felix W; Chekler, Eugene; Garces, Robert; Wolff, Karen C; Riva, Laura; Kirkpatrick, Melanie G; Gebara-Lamb, Amal; McNamara, Case W; Betz, Ulrich A K; Arumugaswami, Vaithilingaraja; Damoiseaux, Robert; Gomperts, Brigitte N

Hydrophobic Eutectic Solvents for Sustainable Bisphenol A Extraction from Water: Screening and Selection Based on Key Performance Criteria

用于从水中可持续提取双酚A的疏水性共熔溶剂:基于关键性能标准的筛选和选择

Carotti, Chiara; Righetti, Grazia Isa C; Mannu, Alberto; Rossetti, Arianna; Riva, Laura; Nicastro, Gloria; Briatico Vangosa, Francesco; Punta, Carlo; Mele, Andrea; Di Pietro, Maria Enrica

Screening of Medicines for Malaria Venture Open Boxes Identifies Potent SARS-CoV‑2 Papain-like Protease (PL(pro)) Inhibitors

疟疾药物筛选项目“开放盒子”发现了强效的SARS-CoV-2木瓜蛋白酶样蛋白酶(PL(pro))抑制剂

Gawriljuk, Victor Oliveira; Noske, Gabriela Dias; Fernandes, Rafaela Sachetto; Nakamura, Aline Minalli; Freire, Marjorie C L C; Godoy, Mariana Ortiz; Bonatto, Vinicius; Chelucci, Rafael; Andricopulo, Adriano; Bakowski, Malina A; Wolff, Karen C; Riva, Laura; Burrows, Jeremy N; Wells, Timothy N C; Laleu, Benoît; Martins, Ronaldo; Souza, Juliano Paula; Arruda, Eurico; Samby, Kirandeep; Laskar, Sujay; Guido, Rafael Victorio Carvalho; Oliva, Glaucius; Godoy, Andre Schutzer

Open Source Repurposing Reveals Broad-Spectrum Antiviral Activity of Diphenylureas.

开源药物再利用揭示了二苯脲的广谱抗病毒活性

Betz Ulrich A K, Garces Robert, Beier Norbert, Lindemann Sven, Wolff Karen C, Riva Laura, Kirkpatrick Melanie G, Gebara-Lamb Amal, McNamara Case W, Damoiseaux Robert, Gomperts Brigitte N, Arumugaswami Vaithilingaraja, Strand MÃ¥rten, Gwon Yongdae, Elofsson Mikael, Evander Magnus

Synthesis and Structure-Activity Relationship of Covalent Inhibitors of SARS-CoV-2 Papain-Like Protease with Antiviral Potency

SARS-CoV-2木瓜蛋白酶样蛋白酶共价抑制剂的合成及构效关系及其抗病毒活性

Rouch, Catherine C; Chatterjee, Arnab K; McCarty, Connor; Song, Lirui; Chu, Alan; Johnson, Kristen; Heacock, Mina; Riva, Laura; McNamara, Case W; Wolff, Karen C; Greene-Cramer, Rebecca; Falco, Anna De; Montelione, Gaetano T; Grabovyi, Gennadii A

Mediastinal staging of nonsmall cell lung cancer: what's new?

非小细胞肺癌纵隔分期:有哪些新进展?

Bradley, Claire; Novoa, Nuria; Riva, Laura; Lampaki, Sophia; Ricciardi, Sara; Rovanias, Michael; Chaabouni, Malek; Turner, Richard; Zachariou, Antonia; Hardavella, Georgia; Navani, Neal

An oral non-covalent non-peptidic inhibitor of SARS-CoV-2 Mpro ameliorates viral replication and pathogenesis in vivo.

SARS-CoV-2 Mpro 的口服非共价非肽抑制剂可改善体内病毒复制和致病性

Zhou Nian E, Tang Su, Bian Xuelin, Parai Maloy K, Krieger Inna V, Flores Armando, Jaiswal Pradeep K, Bam Radha, Wood Jeremy L, Shi Zhe, Stevens Laura J, Scobey Trevor, Diefenbacher Meghan V, Moreira Fernando R, Baric Thomas J, Acharya Arjun, Shin Joonyoung, Rathi Manish M, Wolff Karen C, Riva Laura, Bakowski Malina A, McNamara Case W, Catanzaro Nicholas J, Graham Rachel L, Schultz David C, Cherry Sara, Kawaoka Yoshihiro, Halfmann Peter J, Baric Ralph S, Denison Mark R, Sheahan Timothy P, Sacchettini James C

Discovery of CMX990: A Potent SARS-CoV-2 3CL Protease Inhibitor Bearing a Novel Warhead

CMX990 的发现:一种带有新型弹头的强效 SARS-CoV-2 3CL 蛋白酶抑制剂

Dayan Elshan, N G R; Wolff, Karen C; Riva, Laura; Woods, Ashley K; Grabovyi, Gennadii; Wilson, Katy; Pedroarena, James; Ghorai, Sourav; Nazarian, Armen; Weiss, Frank; Liu, Yuyin; Mazumdar, Wrickban; Song, Lirui; Okwor, Neechi; Malvin, Jacqueline; Bakowski, Malina A; Beutler, Nathan; Kirkpatrick, Melanie G; Gebara-Lamb, Amal; Huang, Edward; Nguyen-Tran, Vân T B; Chi, Victor; Li, Shuangwei; Rogers, Thomas F; McNamara, Case W; Gupta, Anil Kumar; Rahimi, Alireza; Chen, Jian Jeffrey; Joseph, Sean B; Schultz, Peter G; Chatterjee, Arnab K