日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Using the Scaffold of FDA-Approved Drugs with Trypanocidal Activity to Identify New Anti-Trypanosoma cruzi Agents: An In Silico and In Vitro Approach

利用已获FDA批准的具有锥虫杀灭活性的药物骨架来鉴定新的抗克氏锥虫药物:一种计算机模拟和体外方法

Yamamuro, Tadashi; Katoh, Daisuke; Silva, Guilherme Martins; Nishida, Hiroshi; Oikawa, Satoshi; Higuchi, Yusuke; Wang, Dandan; Fujimoto, Masanori; Yoshida, Naofumi; Li, Mark; Shin, Jihoon; Zhao, Zezhou; Yook, Jin-Seon; Sun, Lijun; Kajimura, Shingo; Xie, Qingchao; Liu, Yihui; Zhang, Zhe; Zhang, Hongmin; Xu, Jin; Wang, Yeru; Zhao, Yong; Zhao, Qingxia; Song, Jingyi; Li, Xukai; Zhang, Zhongwei; Xiao, Junsong; Wu, Hua; Huang, Mingquan; Boppana, Sri Harsha; Luke, Naveena; Karuchola, Sravani; Udaikumar, Jahnavi; Mintz, Cyrus David; Zhou, Yaxi; Xu, Dong; Bu, Meichao; Li, Ke; Gao, Lingyu; Pan, Fei; Peng, Wenjun; Chen, Hualei; Tian, Wenli; Lyu, Yipin; Zhang, Jie; Cheng, Chi; Tang, Xue; Huang, Pantian; Liu, Feitong; Hu, Ruibiao; Huppertz, Thom; Wang, Xinyan; Zhou, Peng; Zhang, Xiaojing; Xing, Huizhen; Liu, Huiping; Zhang, Xiaowei; Vázquez-Jiménez, Lenci K; González-González, Alonzo; Delgado-Maldonado, Timoteo; Gómez-Escobedo, Rogelio; Avalos-Navarro, Guadalupe; Moreno-Rodríguez, Adriana; Paz-González, Alma D; Ortiz-Pérez, Eyra; Nogueda-Torres, Benjamín; Rivera, Gildardo

An In Silico and In Vitro Approach Identified Potential Trypanothione Synthetase Inhibitors with Trypanocidal Activity

通过计算机模拟和体外实验方法,鉴定出具有锥虫杀灭活性的潜在锥虫硫合成酶抑制剂。

Gómez-Escobedo, Rogelio; Méndez-Álvarez, Domingo; Paz-González, Alma D; Ortiz-Pérez, Eyra; Vázquez-Jiménez, Lenci K; Martínez-Vázquez, Ana Verónica; Delgado-Maldonado, Timoteo; Quintero-Solano, José M; Vázquez, Citlali; Saavedra, Emma; Avalos-Navarro, Guadalupe; Vázquez, Karina; Rivera, Gildardo; Nogueda-Torres, Benjamín

Identification of Novel Trypanosoma cruzi Cysteine Protease Inhibitors via Ligand-Based Virtual Screening of FDA-Approved Drugs with Trypanocidal Activity

通过基于配体的虚拟筛选方法,从FDA批准的具有锥虫杀灭活性的药物中鉴定新型克氏锥虫半胱氨酸蛋白酶抑制剂

Vázquez-Jiménez, Lenci K; González-González, Alonzo; Delgado-Maldonado, Timoteo; Gómez-Escobedo, Rogelio; Nogueda-Torres, Benjamín; Martínez-Vázquez, Ana Verónica; Ortiz-Pérez, Eyrá; Aguirre-Alvarado, Charmina; Alcántara-Farfán, Verónica; Cordero-Martínez, Joaquín; Rodríguez-Páez, Lorena; Moreno-Rodriguez, Adriana; Rivera, Gildardo

Carotid Intima–Media Thickness and Narrowing in Rheumatoid Arthritis: Impact of Age, Diabetes, and Conventional Risk Factors

类风湿性关节炎患者颈动脉内膜中层厚度和狭窄:年龄、糖尿病和传统危险因素的影响

Ford, Jessie V; Coleman, Eli; de Oliveira, Leonor; Rahm-Knigge, Ryan L; Mark, Kristen P; Vázquez-Jiménez, Lenci K; González-González, Alonzo; Delgado-Maldonado, Timoteo; Gómez-Escobedo, Rogelio; Avalos-Navarro, Guadalupe; Moreno-Rodríguez, Adriana; Paz-González, Alma D; Ortiz-Pérez, Eyra; Nogueda-Torres, Benjamín; Rivera, Gildardo; Almutairi, Fahad F; Alsalah, Jaber H; Alzubaidi, Husam K; Mustafa, Mohammad; Bawazir, Yasser; Bahamdein, Khalid; Balubaid, Hassan; Alnahdi, Haifa; Khashoggi, Khalid; Almutairi, Bander; Shetewi, Shoaa; Alrwaithi, Fahad; Abushaheen, Shadi; Attraji, Dana; Alsaylani, Sara; Alamri, Huda; Abdeen, Rawan; Ahmed, Hamzah H; Khalil, Mohammad

Design, Synthesis, In Vitro and In Silico Biological Evaluation of New Pyridine-2,5-Dicarboxylates Esters Bearing Natural Source Fragments as Anti-Trypanosomatid Agents

设计、合成、体外和计算机生物学评价含天然来源片段的新型吡啶-2,5-二羧酸酯类化合物作为抗锥虫药物

Sánchez-Palestino, Luis M; Moreno-Rodríguez, Adriana; Navarrete-Carriola, Diana V; Martínez-Archundia, Marlet; López-Vargas, Marhian; Argueta-Figueroa, Liliana; Vázquez-Jiménez, Lenci K; Paz-González, Alma D; Ortiz-Pérez, Eyra; Doyle, Michael P; Rivera, Gildardo

Nifuroxazide and 4-Hydroxybenzhydrazone Derivatives as New Antiparasitic (Trypanosoma cruzi and Leishmania mexicana) and Anti-Mycobacterium tuberculosis Agents

硝呋嗪和4-羟基苯甲腙衍生物作为新型抗寄生虫(克氏锥虫和墨西哥利什曼原虫)和抗结核分枝杆菌药物

Delgado-Maldonado, Timoteo; Navarrete-Carriola, Diana V; Vázquez-Jiménez, Lenci K; Paz-González, Alma D; Wan, Baojie; Franzblau, Scott; Mohammed, Othman Mueen; Rodríguez-Páez, Lorena; Aguirre-Alvarado, Charmina; Alcántara-Farfán, Verónica; Cordero-Martínez, Joaquín; Bandyopadhyay, Debasish; Moreno-Rodríguez, Adriana; Rivera, Gildardo

The Arg108Cys Variant of Methylmalonyl-CoA Mutase: Clinical Implications for the Mexican Population Based on Molecular Dynamics and Docking

甲基丙二酰辅酶A变位酶Arg108Cys变体:基于分子动力学和分子对接的墨西哥人群临床意义

Vela-Amieva, Marcela; Delgado-Maldonado, Timoteo; Ortega-Valdez, Enrique; Rivera, Gildardo; López-Velázquez, Gabriel; Fernández-Lainez, Cynthia

In Silico Investigation of TATA-Binding Protein as a Therapeutic Target for Chagas Disease: Insights into FDA Drug Repositioning

利用计算机模拟研究TATA结合蛋白作为恰加斯病治疗靶点:对FDA药物重定位的启示

Gaona-López, Carlos; Méndez-Álvarez, Domingo; Gonzalez-Gonzalez, Alonzo; Avalos-Navarro, Guadalupe; Paz-González, Alma D; Moreno-Rodríguez, Adriana; Nogueda-Torres, Benjamín; Rivera, Gildardo

Repositioning FDA-Approved Sulfonamide-Based Drugs as Potential Carbonic Anhydrase Inhibitors in Trypanosoma cruzi: Virtual Screening and In Vitro Studies

将FDA批准的磺胺类药物重新定位为克氏锥虫潜在碳酸酐酶抑制剂:虚拟筛选和体外研究

Ortiz-Pérez, Eyra; Moreno-Rodríguez, Adriana; Delgado-Maldonado, Timoteo; Ortega-Balleza, Jessica L; González-González, Alonzo; Paz-González, Alma D; Vázquez, Karina; Avalos-Navarro, Guadalupe; Giovannuzzi, Simone; Supuran, Claudiu T; Rivera, Gildardo

In Vitro Evaluation of Esters of Quinoxaline-1,4-di-N-oxide Derivatives as New Antitaeniasis Agents and Their Inhibitory Activity Against Triosephosphate Isomerase

体外评价喹喔啉-1,4-二-N-氧化物衍生物酯类作为新型抗绦虫病药物的活性及其对磷酸丙糖异构酶的抑制活性

Palomares-Alonso, Francisca; González-González, Alonzo; Paz-González, Alma D; Ortiz-Pérez, Eyra; Martínez-Vázquez, Ana Verónica; García-Torres, Itzhel; López-Velázquez, Gabriel; Jung-Cook, Helgi; Rivera, Gildardo