日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification and Validation of an Inhibitor of the Protein Kinases PIM and DYRK.

鉴定和验证蛋白激酶 PIM 和 DYRK 的抑制剂。

Bencze Gyula, Venkataramani Prabhadevi, Elkayam Elad, Rivera Keith D, Garg Ankur, Szabadakai Istvan, Orfi Laszlo, Joshua-Tor Leemor, Pappin Darryl J, Tonks Nicholas K

Identification and Validation of an inhibitor of the protein kinases PIM and DYRK

鉴定和验证蛋白激酶 PIM 和 DYRK 的抑制剂

Bencze, Gyula; Venkataramani, Prabhadevi; Elkayam, Elad; Rivera, Keith D; Garg, Ankur; Szabadkai, Istvan; Orfi, Laszlo; Joshua-Tor, Leemor; Pappin, Darryl; Tonks, Nicholas K

Dietary pro-oxidant therapy by a vitamin K precursor targets PI 3-kinase VPS34 function.

通过维生素 K 前体进行膳食促氧化疗法,可靶向 PI 3-激酶 VPS34 的功能

Swamynathan Manojit M, Kuang Shan, Watrud Kaitlin E, Doherty Mary R, Gineste Charlotte, Mathew Grinu, Gong Grace Q, Cox Hilary, Cheng Eileen, Reiss David, Kendall Jude, Ghosh Diya, Reczek Colleen R, Zhao Xiang, Herzka Tali, Špokaitė Saulė, Dessus Antoine N, Kim Seung Tea, Klingbeil Olaf, Liu Juan, Nowak Dawid G, Alsudani Habeeb, Wee Tse-Luen, Park Youngkyu, Minicozzi Francesca, Rivera Keith, Almeida Ana S, Chang Kenneth, Chakrabarty Ram P, Wilkinson John E, Gimotty Phyllis A, Diermeier Sarah D, Egeblad Mikala, Vakoc Christopher R, Locasale Jason W, Chandel Navdeep S, Janowitz Tobias, Hicks James B, Wigler Michael, Pappin Darryl J, Williams Roger L, Cifani Paolo, Tuveson David A, Laporte Jocelyn, Trotman Lloyd C

Prostate tumor-induced stromal reprogramming generates Tenascin C that promotes prostate cancer metastasis through YAP/TAZ inhibition

前列腺肿瘤诱导的基质重编程产生腱生蛋白C,后者通过抑制YAP/TAZ促进前列腺癌转移。

Lee, Yu-Chen; Lin, Song-Chang; Yu, Guoyu; Zhu, Ming; Song, Jian H; Rivera, Keith; Pappin, Darryl J; Logothetis, Christopher J; Panaretakis, Theocharis; Wang, Guocan; Yu-Lee, Li-Yuan; Lin, Sue-Hwa

Tryp-N: A Thermostable Protease for the Production of N-terminal Argininyl and Lysinyl Peptides

Tryp-N:一种用于生产N端精氨酰肽和赖氨酰肽的耐热蛋白酶

Wilson, John P; Ipsaro, Jonathan J; Del Giudice, Samantha N; Turna, Nikita Saha; Gauss, Carla M; Dusenbury, Katharine H; Marquart, Krisann; Rivera, Keith D; Pappin, Darryl J

SARS-CoV-2 infected cells present HLA-I peptides from canonical and out-of-frame ORFs

SARS-CoV-2感染细胞会呈递来自经典开放阅读框和移码开放阅读框的HLA-I肽。

Weingarten-Gabbay, Shira; Klaeger, Susan; Sarkizova, Siranush; Pearlman, Leah R; Chen, Da-Yuan; Bauer, Matthew R; Taylor, Hannah B; Conway, Hasahn L; Tomkins-Tinch, Christopher H; Finkel, Yaara; Nachshon, Aharon; Gentili, Matteo; Rivera, Keith D; Keskin, Derin B; Rice, Charles M; Clauser, Karl R; Hacohen, Nir; Carr, Steven A; Abelin, Jennifer G; Saeed, Mohsan; Sabeti, Pardis C

The glycan CA19-9 promotes pancreatitis and pancreatic cancer in mice

糖链CA19-9可促进小鼠胰腺炎和胰腺癌的发生。

Engle, Dannielle D; Tiriac, Hervé; Rivera, Keith D; Pommier, Arnaud; Whalen, Sean; Oni, Tobiloba E; Alagesan, Brinda; Lee, Eun Jung; Yao, Melissa A; Lucito, Matthew S; Spielman, Benjamin; Da Silva, Brandon; Schoepfer, Christina; Wright, Kevin; Creighton, Brianna; Afinowicz, Lauren; Yu, Kenneth H; Grützmann, Robert; Aust, Daniela; Gimotty, Phyllis A; Pollard, Katherine S; Hruban, Ralph H; Goggins, Michael G; Pilarsky, Christian; Park, Youngkyu; Pappin, Darryl J; Hollingsworth, Michael A; Tuveson, David A

DPM-1001 decreased copper levels and ameliorated deficits in a mouse model of Wilson's disease

DPM-1001降低了小鼠威尔逊病模型中的铜水平并改善了其功能缺陷。

Krishnan, Navasona; Felice, Christy; Rivera, Keith; Pappin, Darryl J; Tonks, Nicholas K

Efficient Reassignment of a Frequent Serine Codon in Wild-Type Escherichia coli

高效重分配野生型大肠杆菌中频繁出现的丝氨酸密码子

Ho, Joanne M; Reynolds, Noah M; Rivera, Keith; Connolly, Morgan; Guo, Li-Tao; Ling, Jiqiang; Pappin, Darryl J; Church, George M; Söll, Dieter

BET Bromodomain Inhibition Suppresses the Function of Hematopoietic Transcription Factors in Acute Myeloid Leukemia

BET溴结构域抑制剂抑制急性髓系白血病中造血转录因子的功能

Roe, Jae-Seok; Mercan, Fatih; Rivera, Keith; Pappin, Darryl J; Vakoc, Christopher R