日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Thieno[2,3- d]pyrimidine-2,4(1 H,3 H)-dione Derivative Inhibits d-Dopachrome Tautomerase Activity and Suppresses the Proliferation of Non-Small Cell Lung Cancer Cells

噻吩并[2,3-d]嘧啶-2,4(1H,3H)-二酮衍生物抑制d-多巴色素互变异构酶活性并抑制非小细胞肺癌细胞增殖

Zhangping Xiao, Angelina Osipyan, Shanshan Song, Deng Chen, Reinder A Schut, Ronald van Merkerk, Petra E van der Wouden, Robbert H Cool, Wim J Quax, Barbro N Melgert, Gerrit J Poelarends, Frank J Dekker

D-dopachrome tautomerase contributes to lung epithelial repair via atypical chemokine receptor 3-dependent Akt signaling

D-多巴色素互变酶通过非典型趋化因子受体3依赖的Akt信号通路促进肺上皮修复

Shanshan Song ,Bin Liu ,Habibie Habibie ,Jelle van den Bor ,Martine J Smit ,Reinoud Gosens ,Xinhui Wu ,Corry-Anke Brandsma ,Robbert H Cool ,Hidde J Haisma ,Gerrit J Poelarends ,Barbro N Melgert

Proteolysis Targeting Chimera (PROTAC) for Macrophage Migration Inhibitory Factor (MIF) Has Anti-Proliferative Activity in Lung Cancer Cells

针对巨噬细胞移动抑制因子 (MIF) 的蛋白水解靶向嵌合体 (PROTAC) 在肺癌细胞中具有抗增殖活性

Zhangping Xiao, Shanshan Song, Deng Chen, Ronald van Merkerk, Petra E van der Wouden, Robbert H Cool, Wim J Quax, Gerrit J Poelarends, Barbro N Melgert, Frank J Dekker

7-Hydroxycoumarins Are Affinity-Based Fluorescent Probes for Competitive Binding Studies of Macrophage Migration Inhibitory Factor

7-羟基香豆素是基于亲和力的荧光探针,用于巨噬细胞迁移抑制因子的竞争性结合研究

Zhangping Xiao, Deng Chen, Shanshan Song, Ramon van der Vlag, Petra E van der Wouden, Ronald van Merkerk, Robbert H Cool, Anna K H Hirsch, Barbro N Melgert, Wim J Quax, Gerrit J Poelarends, Frank J Dekker

Creation of RANKL mutants with low affinity for decoy receptor OPG and their potential anti-fibrosis activity

构建对诱饵受体 OPG 具有低亲和力的 RANKL 突变体及其潜在的抗纤维化活性

Yizhou Wang, Timo Michiels, Rita Setroikromo, Ronald van Merkerk, Robbert H Cool, Wim J Quax

Heightened JNK Activation and Reduced XIAP Levels Promote TRAIL and Sunitinib-Mediated Apoptosis in Colon Cancer Models

在结肠癌模型中,JNK 活性增强和 XIAP 水平降低促进 TRAIL 和舒尼替尼介导的细胞凋亡

Devalingam Mahalingam, Jennifer S Carew, Claudia M Espitia, Robbert H Cool, Francis J Giles, Steven de Jong, Steffan T Nawrocki

PvdP is a tyrosinase that drives maturation of the pyoverdine chromophore in Pseudomonas aeruginosa

PvdP 是一种酪氨酸酶,可促进铜绿假单胞菌中绿脓杆菌发色团的成熟

Pol Nadal-Jimenez, Gudrun Koch, Carlos R Reis, Remco Muntendam, Hans Raj, C Margot Jeronimus-Stratingh, Robbert H Cool, Wim J Quax

Kinetics in signal transduction pathways involving promiscuous oligomerizing receptors can be determined by receptor specificity: apoptosis induction by TRAIL

涉及混杂寡聚化受体的信号转导途径的动力学可以通过受体特异性来确定:TRAIL 诱导细胞凋亡

Eva Szegezdi, Almer M van der Sloot, Devalingam Mahalingam, Lynda O'Leary, Robbert H Cool, Inés G Muñoz, Guillermo Montoya, Wim J Quax, Steven de Jong, Afshin Samali, Luis Serrano

Unraveling the binding mechanism of trivalent tumor necrosis factor ligands and their receptors

揭示三价肿瘤坏死因子配体与其受体的结合机制

Carlos R Reis, Aart H G van Assen, Wim J Quax, Robbert H Cool

Targeting AML through DR4 with a novel variant of rhTRAIL

利用 rhTRAIL 的新变体通过 DR4 靶向 AML

Eva Szegezdi, Carlos R Reis, Almer M van der Sloot, Alessandro Natoni, Aoife O'Reilly, Janice Reeve, Robbert H Cool, Michael O'Dwyer, Steven Knapper, Luis Serrano, Wim J Quax, Afshin Samali