日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting β-catenin: PROTACs and precision degraders for Wnt-driven cancers

靶向β-catenin:PROTACs和精准降解剂治疗Wnt驱动型癌症

Trapani, Jonathan; Caroland, Kailey P; Ahmed, Yashi; Robbins, David J; Weiss, Vivian L; Lee, Ethan

The TRIP12 E3 ligase induces SWI/SNF component BRG1-β-catenin interaction to promote Wnt signaling.

TRIP12 E3 连接酶诱导 SWI/SNF 成分 BRG1-β-catenin 相互作用,从而促进 Wnt 信号传导

Kassel Sara, Yuan Kai, Bunnag Nawat, Neitzel Leif R, Lu Wenhui, Schwarzkopf Anna, Maines Benjamin, Loberg Matthew A, Xu George, Adams Amber, McCray Andrew D, Cho Alex, Rockouski Mary, Orton Gemma, Goldsmith Lily, Aronno Md Mubtaseem Ahnaf, Spencer Zachary T, Khan Omar M, Ye Fei, Williams Charles, Lebensohn Andres M, Rohatgi Rajat, Wang Xiaofeng, Weiss Vivian L, Hong Charles C, Kettenbach Arminja N, Robbins David J, Ahmed Yashi, Lee Ethan

Lipid peroxidation products induce carbonyl stress, mitochondrial dysfunction, and cellular senescence in human and murine cells

脂质过氧化产物会诱发人类和鼠类细胞的羰基应激、线粒体功能障碍和细胞衰老

T Blake Monroe, Ann V Hertzel, Deborah M Dickey, Thomas Hagen, Simon Vergara Santibanez, Islam A Berdaweel, Catherine Halley, Patrycja Puchalska, Ethan J Anderson, Christina D Camell, Paul D Robbins, David A Bernlohr

Wnt signaling inhibits casein kinase 1α activity by modulating its interaction with protein phosphatase 2A.

Wnt信号通过调节酪蛋白激酶1α与蛋白磷酸酶2A的相互作用来抑制酪蛋白激酶1α的活性。

Shen Chen, Lu Wenhui, Merugu Siva B, Bharti Aradhana, Afify Said M, Schnitkey Lauren, Wynn Daniel T, Yang Fan, Rohwetter Thomas M, Nayak Anmada, Bunnag Nawat, Cywiak Carolina, Tang Hsin-Yao, Harris Brent T, Albanese Christopher, Ihemelandu Chukwuemeka, Cobb Melanie H, Kettenbach Arminja, Lee Ethan, Ahmed Yashi, Robbins David J

Wnt signalosomes: What we know that we do not know

Wnt信号体:我们已知但未知的部分

Hartmann, Heather; Siddiqui, Ghalia Saad; Bryant, Jamal; Robbins, David J; Weiss, Vivian L; Ahmed, Yashi; Lee, Ethan

RAC1 Regulates Shh-Medulloblastoma Growth via GLI-Mediated Transcription

RAC1通过GLI介导的转录调控Shh-髓母细胞瘤的生长

Jangde, Nitish; Lee, Mi Hye; Ruiz, Luz; Egan, Isabelle; Jermakowicz, Anna M; Wynn, Daniel; Goka, Erik; Lippman, Marc; Robbins, David J; Ayad, Nagi G

DIPG-68. FLAG-003, A NOVEL, DUAL-ACTION THERAPEUTIC, DEMONSTRATES IN-VITRO ACTIVITY AGAINST DIFFUSE INTRINSIC PONTINE GLIOMA (DIPG)

DIPG-68. FLAG-003,一种新型双效疗法,在体外显示出对弥漫性内生性脑桥胶质瘤(DIPG)的活性。

Vishakantegowda, Avinash G; Hwang, Dasom; Chakrasali, Prashant; Jung, Eunhye; Lee, Joo-Youn; Shin, Jin Soo; Jung, Young-Sik; Alahdal, Murad; Perera, Ranjan J; Chaleff, Stanley; Gerwin, Roselyn; Wolfrum, Lee; Bokat, Pamela; Kastle, Nadav; Amal, Mohamad Yanuar; Rahmartani, Ludi Dhyani; Susanto, Eka; Davenport, Alexander J; Lertsumitkul, Leesa; Cross, Ryan S; Jenkins, Misty R; Levin, Jared; Rosenberg, Nathan; Tsao, Elaine; Liapodimitri, Athanasia; Lunsford, Kayleigh; Tetens, Ashley R; Craig-Schwartz, Jordyn; Vesuna, Farhad; Raman, Venu; Koldobskiy, Michael A; Ashraf, Nader; Kofide, Amani Al; Arabi, Tarek; Sabbah, Belal; Aboian, Mariam; Ouban, Abderrahman; Matson, Kathryn; Corr, Gwendolyn; Maack, Lennart; Kresbach, Catena; Neumann, Julia; Tischendorf, Jacqueline; Wefers, Annika; Seegerer, Philipp; Schüller, Ulrich; Schlaefer, Alexander; Bockmayr, Michael; Donson, Andrew M; Griesinger, Andrea M; Calzadilla, Annaliese; Amani, Vladimir; Grimaldo, Enrique; Foreman, Nicholas K; Rizzo, Deborah R; Hayes, Melissa; Blount, Nicola; Robinson, Louise; Reynolds, Gabrielle; Ryles, Jade; Lyons, Nicole; Ward, Lisa; Katsushima, Keisuke; Joshi, Kandarp; Yuan, Menglang; Batish, Mona; Stapleton, Stacie; Jallo, George; Seal, Sudipta; Taylor, Michael D; Wechsler-Reya, Rober J; Eberhart, Charles G; Perera, Ranjan J; McAndrew, Rachel; Laughlin, Elizabeth; Page, Joanne; Paisley, Helen; Howat, Angela; Coyle, Paul; Jangde, Nitish; Wynn, Daniel; Egan, Isabelle; Robbins, David; Ayad, Nagi; Fitzgerald, Caroline; Phelan, Alison; Chilukuri, Akanksha; Pomaville, Monica; Halbert, Matthew; He, Chaun; Agnihotri, Sameer; Li, Daphne; Stellpflug, Wendy; Romanski, Kathy; Speck, Stacy; Saratsis, Amanda; Bhatia, Sonam; Quinn, Thomas; Ligon, Keith L; Bandopadhayay, Pratiti; Warren, Katherine

Enhancing precision in colorectal cancer surgery: development of an LGR5-targeting RSPO1 peptide mimetic as a contrast agent for intraoperative fluorescence molecular imaging.

提高结直肠癌手术的精准度:开发靶向 LGR5 的 RSPO1 肽模拟物作为术中荧光分子成像的对比剂

Parasido Erika, Ribeiro Patricia, Chingle Ramesh M, Rohwetter Thomas, Gupta Nikita, Avetian George, Bladelli Elisa, Pierobon Mariaelena, Chen Yu, Tang Qinggong, Schnermann Martin, Rodriguez Olga, Robbins David, Burke Terrence R Jr, Albanese Chris, Ihemelandu Chukwuemeka

Exploring the role of casein kinase 1α splice variants across cancer cell lines.

探索酪蛋白激酶 1α 剪接变体在癌细胞系中的作用

Meléndez Ricardo A, Wynn Daniel T, Merugu Siva Bharath, Singh Prerna, Kaplan Kenton P, Robbins David J

CNSC-17. WHOLE-BRAIN SPECTRAL CHANGE IN GLIOBLASTOMA PATIENTS: ASSOCIATIONS WITH CLINICAL COMORBIDITIES AND OVERALL SURVIVAL

CNSC-17. 胶质母细胞瘤患者全脑频谱变化:与临床合并症和总生存期的关联

Choi, In-Young; Wang, Wen-Tung; Kim, Bhumsoo; Hur, Junguk; Robbins, David C; Jang, Dae-Gyu; Savelieff, Masha G; Feldman, Eva L; Lee, Phil; Park, Ki Yun; Snyder, Abraham; Olufawo, Michael; Trevino, Gabriel; Luckett, Patrick; Lamichhane, Bidhan; Xie, Tao; Lee, John; Shimony, Joshua; Leuthardt, Eric