日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Binding of small molecules at the P-stalk site of ricin A subunit trigger conformational changes that extend into the active site.

小分子与蓖麻毒素 A 亚基 P 茎位点的结合会引发构象变化,进而延伸至活性位点

McLaughlin John E, Rudolph Michael J, Dutta Arkajyoti, Li Xiao-Ping, Tsymbal Anastasiia M, Chen Yang, Bhattacharya Shibani, Algava Benjamin, Goger Michael, Roberge Jacques Y, Tumer Nilgun E

A FtsZ inhibitor-acinetobactin conjugate with enhanced cellular uptake in Acinetobacter baumannii acts synergistically in combination with PBP3-targeting antibiotics

一种FtsZ抑制剂-不动杆菌素偶联物可增强鲍曼不动杆菌的细胞摄取,并与靶向PBP3的抗生素协同作用。

Bryan, Eric J; Szekely, Zoltan; Wang, Yuxuan; Fan, Huizhou; Moynié, Lucile; Roberge, Jacques Y; Pilch, Daniel S

Fragment Screening to Identify Inhibitors Targeting Ribosome Binding of Shiga Toxin 2

利用片段筛选鉴定靶向志贺毒素2核糖体结合的抑制剂

Rudolph, Michael J; Tsymbal, Anastasiia M; Dutta, Arkajyoti; Davis, Simon A; Algava, Benjamin; Roberge, Jacques Y; Tumer, Nilgun E; Li, Xiao-Ping

The Anticancer Drug Bleomycin Shows Potent Antifungal Activity by Altering Phospholipid Biosynthesis

抗癌药物博来霉素通过改变磷脂生物合成而表现出强大的抗真菌活性。

Pokharel, Mona; Konarzewska, Paulina; Roberge, Jacques Y; Han, Gil-Soo; Wang, Yina; Carman, George M; Xue, Chaoyang