日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Multi-Omics Approach Reveals Enrichment in Metabolites Involved in the Regulation of the Glutathione Pathway in LIN28B-Dependent Cancer Cells

多组学方法揭示 LIN28B 依赖性癌细胞中参与调节谷胱甘肽途径的代谢物的富集

Matteo Stocchero, Diana Corallo, Silvia Bresolin, Marcella Pantile, Paola Pirillo, Roberta Bortolozzi, Sara Menegazzo, Daniele Boso, Giampietro Viola, Eugenio Baraldi, Alessandra Biffi, Giuseppe Giordano, Sanja Aveic

Molecular and functional profiling of chemotolerant cells unveils nucleoside metabolism-dependent vulnerabilities in medulloblastoma

化学耐受细胞的分子和功能分析揭示了髓母细胞瘤中核苷代谢依赖性的脆弱性

Elena Mariotto #, Elena Rampazzo #, Roberta Bortolozzi #, Fatlum Rruga, Ilaria Zeni, Lorenzo Manfreda, Chiara Marchioro, Martina Canton, Alice Cani, Ruben Magni, Alessandra Luchini, Silvia Bresolin, Giampietro Viola #, Luca Persano #

Design, synthesis, and biological investigation of selective human carbonic anhydrase II, IX, and XII inhibitors using 7-aryl/heteroaryl triazolopyrimidines bearing a sulfanilamide scaffold

使用带有磺胺支架的 7-芳基/杂芳基三唑并嘧啶设计、合成并进行选择性人类碳酸酐酶 II、IX 和 XII 抑制剂的生物学研究

Romeo Romagnoli, Tiziano De Ventura, Stefano Manfredini, Erika Baldini, Claudiu T Supuran, Alessio Nocentini, Andrea Brancale, Roberta Bortolozzi, Lorenzo Manfreda, Giampietro Viola

Synthesis and Biological Evaluation of Highly Active 7-Anilino Triazolopyrimidines as Potent Antimicrotubule Agents

高活性 7-苯胺基三唑并嘧啶作为强效抗微管剂的合成及生物学评价

Paola Oliva, Romeo Romagnoli, Barbara Cacciari, Stefano Manfredini, Chiara Padroni, Andrea Brancale, Salvatore Ferla, Ernest Hamel, Diana Corallo, Sanja Aveic, Noemi Milan, Elena Mariotto, Giampietro Viola, Roberta Bortolozzi

Histone Deacetylase Inhibitors Impair Glioblastoma Cell Motility and Proliferation

组蛋白去乙酰化酶抑制剂损害胶质母细胞瘤细胞的运动能力和增殖

Elena Rampazzo, Lorenzo Manfreda, Silvia Bresolin, Alice Cani, Elena Mariotto, Roberta Bortolozzi, Alessandro Della Puppa, Giampietro Viola, Luca Persano

Ecdysteroid Derivatives that Reverse P-Glycoprotein-Mediated Drug Resistance

逆转 P-糖蛋白介导的耐药性的蜕皮类固醇衍生物

Roberta Bortolozzi, Andrea Luraghi, Elena Mattiuzzo, Alessandro Sacchetti, Alessandra Silvani, Giampietro Viola

AKR1C enzymes sustain therapy resistance in paediatric T-ALL

AKR1C 酶维持儿童 T-ALL 的治疗耐药性

Roberta Bortolozzi, Silvia Bresolin, Elena Rampazzo, Maddalena Paganin, Francesca Maule, Elena Mariotto, Daniele Boso, Sonia Minuzzo, Valentina Agnusdei, Giampietro Viola, Geertruy Te Kronnie, Giovanni Cazzaniga, Giuseppe Basso, Luca Persano

Targeting tubulin polymerization by novel 7-aryl-pyrroloquinolinones: Synthesis, biological activity and SARs

新型 7-芳基吡咯喹啉酮靶向微管蛋白聚合:合成、生物活性和 SAR

Roberta Bortolozzi, Elena Mattiuzzo, Matteo Dal Pra, Mattia Sturlese, Stefano Moro, Ernest Hamel, Davide Carta, Giampietro Viola, Maria Grazia Ferlin

Synthesis, structure-activity relationships and biological evaluation of 7-phenyl-pyrroloquinolinone 3-amide derivatives as potent antimitotic agents

7-苯基吡咯喹啉酮 3-酰胺衍生物作为强效抗有丝分裂剂的合成、构效关系及生物学评价

Davide Carta, Roberta Bortolozzi, Mattia Sturlese, Veronica Salmaso, Ernest Hamel, Giuseppe Basso, Laura Calderan, Luigi Quintieri, Stefano Moro, Giampietro Viola, Maria Grazia Ferlin

Design, synthesis, crystallization and biological evaluation of new symmetrical biscationic compounds as selective inhibitors of human Choline Kinase α1 (ChoKα1)

作为人类胆碱激酶 α1 (ChoKα1) 选择性抑制剂的新型对称双阳离子化合物的设计、合成、结晶和生物学评价

Santiago Schiaffino-Ortega, Eleonora Baglioni, Elena Mariotto, Roberta Bortolozzi, Lucía Serrán-Aguilera, Pablo Ríos-Marco, M Paz Carrasco-Jimenez, Miguel A Gallo, Ramon Hurtado-Guerrero, Carmen Marco, Giuseppe Basso, Giampietro Viola, Antonio Entrena, Luisa Carlota López-Cara