日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Small molecule screening identifies cytotoxic endoplasmic reticulum-associated degradation inhibitors in multiple myeloma

小分子筛选在多发性骨髓瘤中鉴定出细胞毒性内质网相关降解抑制剂

Kropp, Erin M; Matono, Sho; Wang, Olivia Y; Robida, Aaron M; Kandarpa, Malathi; Grant, Jineigh L; Oleson, Bryndon J; Alt, Andrew; Talpaz, Moshe; Pianko, Matthew J; Li, Qing

A Metabolism-Informed Neural Network Identifies Pathways Influencing the Potency and Toxicity of Antimicrobial Combinations

基于代谢信息的神经网络识别影响抗菌药物组合效力和毒性的通路

Arora, Harkirat Singh; Lev, Katherine; Robida, Aaron; Velmurugan, Ramraj; Chandrasekaran, Sriram

Identification of a TNIK-CDK9 Axis as a Targetable Strategy for Platinum-Resistant Ovarian Cancer.

确定 TNIK-CDK9 轴作为铂耐药卵巢癌的靶向治疗策略

Puleo Noah, Ram Harini, Dziubinski Michele L, Carvette Dylan, Teitel Jessica, Sekhar Sreeja C, Bedi Karan, Robida Aaron, Nakashima Michael M, Farsinejad Sadaf, Iwanicki Marcin, Senkowski Wojciech, Ray Arpita, Bollerman Thomas J, Dunbar James, Richardson Peter, Taddei Andrea, Hudson Chantelle, DiFeo Analisa

Pan-cancer Myc modulator that targets Myc-α-tubulin interaction to drive selective mitotic catastrophe

一种靶向Myc-α-微管蛋白相互作用以驱动选择性有丝分裂灾难的泛癌Myc调节剂

Teitel, Jessica; Farah, Margaret; Dziubinski, Michele L; Lee, Pil; White, Andrew; Sobeck, Alexander; Colina, Jose; Takyi-Williams, John; Wen, Bo; Nurmemmedov, Elmar; Babic, Ivan; Monteiro da Rocha, Andre; Bedi, Karan; Robida, Aaron; McIntyre, Grace; Hotta, Takashi; Lin, Yinzhi; Sekhar, Sreeja C; Ohi, Ryoma; DiFeo, Analisa

Identification of Omaveloxolone as An Endoplasmic Reticulum Associated Degradation Inhibitor That Induces Early Apoptotic Signaling in Multiple Myeloma

鉴定出奥马维洛酮是一种内质网相关降解抑制剂,可诱导多发性骨髓瘤早期凋亡信号传导

Kropp, Erin M; Matono, Sho; Wang, Olivia Y; Robida, Aaron M; Kandarpa, Malathi; Grant, Jineigh L; Oleson, Bryndon J; Alt, Andrew; Talpaz, Moshe; Pianko, Matthew; Li, Qing

A mechanistic neural network model predicts both potency and toxicity of antimicrobial combination therapies

一种基于机制的神经网络模型可以预测抗菌联合疗法的效力和毒性。

Arora, Harkirat Singh; Lev, Katherine; Robida, Aaron; Velmurugan, Ramraj; Chandrasekaran, Sriram

Structure-Activity relationship of 1-(Furan-2ylmethyl)Pyrrolidine-Based Stimulation-2 (ST2) inhibitors for treating graft versus host disease

1-(呋喃-2-基甲基)吡咯烷类刺激-2 (ST2) 抑制剂治疗移植物抗宿主病的构效关系

Yuan, Xinrui; Jiang, Hua; Fu, Denggang; Robida, Aaron; Rajanayake, Krishani; Yuan, Hebao; Wen, Bo; Sun, Duxin; Watch, Brennan T; Chinnaswamy, Krishnapriya; Stuckey, Jeanne A; Paczesny, Sophie; Rech, Jason C; Yang, Chao-Yie

Characterisation of an epigenetically altered CD4(+) CD28(+) Kir(+) T cell subset in autoimmune rheumatic diseases by multiparameter flow cytometry

利用多参数流式细胞术对自身免疫性风湿病中表观遗传改变的CD4(+)CD28(+)Kir(+)T细胞亚群进行表征

Strickland, Faith M; Patel, Dipak; Khanna, Dinesh; Somers, Emily; Robida, Aaron M; Pihalja, Michael; Swartz, Richard; Marder, Wendy; Richardson, Bruce