Discovery of small molecules and a druggable groove that regulate DNA binding and release of the AP-1 transcription factor ΔFOSB
发现能够调控AP-1转录因子ΔFOSB的DNA结合和释放的小分子和可成药沟槽
期刊:Journal of Biological Chemistry
影响因子:3.9
doi:10.1016/j.jbc.2025.111080
McNeme, Sean; Yim, Yun Young; Kumar, Ashwani; Li, Yi; Hughes, Brandon; St Romain, Corey Peyton; Aglyamova, Galina; Chen, Jianping; Nguyen, Nghi D; Fan, Shanghua; Stephens, Gabriel S; Zhao, Wen-Ning; Kruzshak, Samantha; Estill, Molly; Brener, Corrine; Tofani, Solange; Kumar, Anil; Chen, Earnest P; Takatka, Nadeen; Robison, Alfred J; Chen, Haiying; Powell, Reid T; Haggarty, Stephen J; Stephan, Clifford; Nestler, Eric J; Chin, Jeannie; Machius, Mischa; Zhou, Jia; Rudenko, Gabby