Aminomethyl-Derived Beta Secretase (BACE1) Inhibitors: Engaging Gly230 without an Anilide Functionality
氨甲基衍生的β-分泌酶(BACE1)抑制剂:无需苯胺官能团即可与Gly230结合
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.6b01451
Butler, Christopher R; Ogilvie, Kevin; Martinez-Alsina, Luis; Barreiro, Gabriela; Beck, Elizabeth M; Nolan, Charles E; Atchison, Kevin; Benvenuti, Eric; Buzon, Leanne; Doran, Shawn; Gonzales, Cathleen; Helal, Christopher J; Hou, Xinjun; Hsu, Mei-Hui; Johnson, Eric F; Lapham, Kimberly; Lanyon, Lorraine; Parris, Kevin; O'Neill, Brian T; Riddell, David; Robshaw, Ashley; Vajdos, Felix; Brodney, Michael A