Leveraging Targeted Protein Degradation for G Protein-Coupled Receptors: The Development of CCR2 Molecular Degraders
利用靶向蛋白降解技术调控G蛋白偶联受体:CCR2分子降解剂的开发
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c02920
Essa, Khaled; Ortiz Zacarías, Natalia V; Roth, Sascha; Xin, Bo-Tao; de Winter, Sabine; van der Horst, Cas; Bleijs, Bente; de Heiden, Richard A; Voulgaraki, Rodanthi; Neubert, Elsa; Ovaa, Huib; Danen, Erik H J; Mulder, Monique P C; Moreau, Kevin; van der Es, Daan; Heitman, Laura H