日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting PTPN22 at Nonorthosteric Binding SitesA Fragment Approach

靶向 PTPN22 的非正构结合位点——片段策略

Di Lello, Paola; Wells, Marta M; Davis, Ben; Daniels, Zoe; Garner, Thomas P; Gazzard, Lewis; Harris, Richard; Hubbard, Roderick E; Landry, Matthew L; Martin, Bryan; Morgan, Jacob L W; Patapoff, Alexander; Simmonite, Heather; Skelton, Nicholas; Ultsch, Mark; Walters, Benjamin T; Wu, Ping; Dimitrova, Yoana N; Huard, Kim

Design, modular synthesis and screening of 58 shape-diverse 3-D fragments

设计、模块化合成和筛选58种形状各异的三维片段

Downes, Thomas D; Jones, S Paul; Firth, James D; Darby, John F; Gilio, Amelia K; Klein, Hanna F; Wang, Xinyu; Blakemore, David C; De Fusco, Claudia; Roughley, Stephen D; Vidler, Lewis R; Whatton, Maria Ann; Woolford, Alison J-A; Wrigley, Gail L; Hubbard, Roderick E; Wu, Liang; Davies, Gideon J; O'Brien, Peter

Characterization of Y chromosome diversity in newfoundland and labrador: evidence for a structured founding population

纽芬兰和拉布拉多Y染色体多样性的特征:结构化创始群体的证据

Zurel, Heather; Bhérer, Claude; Batten, Ryan; MacMillan, Margaret E; Demiriz, Sedat; Mirhendi, Sadra; Gilbert, Edmund; Cavalleri, Gianpiero L; Leach, Richard A; Scott, Roderick E M; Mugford, Gerald; Randhawa, Ranjit; Symington, Alison L; Stephens, J Claiborne; Phillips, Michael S

Altered immunometabolic response to fasting in humans living with obesity.

肥胖人群禁食后免疫代谢反应的改变

Neudorf Helena, Sandilands Roderick E, Ursel Spencer, Shaba Hillary, Barg Darren, Tsusaka Takeshi, Moya-Garzón María Dolores, Vaz Erica, Schimweg Patricia, Goldberg Emily L, Long Jonathan Z, Krüger Karsten, Islam Hashim, Little Jonathan P

Prevalence and Determinants of Antenatal Depression Risk Among Urban Women Seeking Antenatal Clinical Care at a District Hospital in Ghana

加纳某地区医院就诊的城市妇女产前抑郁症风险的患病率及决定因素

Adarkwa, Opei Kwafo; Opoku, Douglas Aninng; Larsen-Reindorf, Roderick E; Owusu-Dabo, Ellis; Boamah, Benedicta; Adarkwa, Magdalene; Obirikorang, Christian; Nartey, Yvonne A; Adjei, Timothy Kwabena; Mohammed, Aliyu

The Newfoundland and Labrador mosaic founder population descends from an Irish and British diaspora from 300 years ago

纽芬兰和拉布拉多岛的创始人口构成多元,其祖先是300年前从爱尔兰和英国移民而来。

Gilbert, Edmund; Zurel, Heather; MacMillan, Margaret E; Demiriz, Sedat; Mirhendi, Sadra; Merrigan, Michael; O'Reilly, Seamus; Molloy, Anne M; Brody, Lawrence C; Bodmer, Walter; Leach, Richard A; Scott, Roderick E M; Mugford, Gerald; Randhawa, Ranjit; Stephens, J Claiborne; Symington, Alison L; Cavalleri, Gianpiero L; Phillips, Michael S

A covalent fragment-based strategy targeting a novel cysteine to inhibit activity of mutant EGFR kinase

一种基于共价片段的策略,靶向一种新型半胱氨酸,以抑制突变型EGFR激酶的活性。

Kuki, Naoki; Walmsley, David L; Kanai, Kazuo; Takechi, Sho; Yoshida, Masao; Murakami, Ryo; Takano, Kohei; Tominaga, Yuichi; Takahashi, Mizuki; Ito, Shuichiro; Nakao, Naoki; Angove, Hayley; Baker, Lisa M; Carter, Edward; Dokurno, Pawel; Le Strat, Loic; Macias, Alba T; Molyneaux, Carrie-Anne; Murray, James B; Surgenor, Allan E; Hamada, Tomoaki; Hubbard, Roderick E

Side-on Coordination in Isostructural Nitrous Oxide and Carbon Dioxide Complexes of Nickel

镍的同构一氧化二氮和二氧化碳配合物中的侧向配位

Puerta Lombardi, Braulio M; Gendy, Chris; Gelfand, Benjamin S; Bernard, Guy M; Wasylishen, Roderick E; Tuononen, Heikki M; Roesler, Roland

Fragment-Derived Selective Inhibitors of Dual-Specificity Kinases DYRK1A and DYRK1B

片段衍生的双特异性激酶 DYRK1A 和 DYRK1B 选择性抑制剂

David Lee Walmsley, James B Murray, Pawel Dokurno, Andrew J Massey, Karen Benwell, Andrea Fiumana, Nicolas Foloppe, Stuart Ray, Julia Smith, Allan E Surgenor, Thomas Edmonds, Didier Demarles, Mike Burbridge, Francisco Cruzalegui, Andras Kotschy, Roderick E Hubbard

P-Rex1 Controls Sphingosine 1-Phosphate Receptor Signalling, Morphology, and Cell-Cycle Progression in Neuronal Cells

P-Rex1 控制神经元细胞中的鞘氨醇 1-磷酸受体信号传导、形态和细胞周期进程

Elizabeth Hampson, Elpida Tsonou, Martin J Baker, David C Hornigold, Roderick E Hubbard, Andrew Massey, Heidi C E Welch