日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fragment-Derived Selective Inhibitors of Dual-Specificity Kinases DYRK1A and DYRK1B

片段衍生的双特异性激酶 DYRK1A 和 DYRK1B 选择性抑制剂

David Lee Walmsley, James B Murray, Pawel Dokurno, Andrew J Massey, Karen Benwell, Andrea Fiumana, Nicolas Foloppe, Stuart Ray, Julia Smith, Allan E Surgenor, Thomas Edmonds, Didier Demarles, Mike Burbridge, Francisco Cruzalegui, Andras Kotschy, Roderick E Hubbard

P-Rex1 Controls Sphingosine 1-Phosphate Receptor Signalling, Morphology, and Cell-Cycle Progression in Neuronal Cells

P-Rex1 控制神经元细胞中的鞘氨醇 1-磷酸受体信号传导、形态和细胞周期进程

Elizabeth Hampson, Elpida Tsonou, Martin J Baker, David C Hornigold, Roderick E Hubbard, Andrew Massey, Heidi C E Welch

Rapid optimisation of fragments and hits to lead compounds from screening of crude reaction mixtures

通过粗反应混合物的筛选快速优化片段并筛选出先导化合物

Lisa M Baker #, Anthony Aimon #, James B Murray, Allan E Surgenor, Natalia Matassova, Stephen D Roughley, Patrick M Collins, Tobias Krojer, Frank von Delft, Roderick E Hubbard

Fragment-derived modulators of an industrial β-glucosidase

工业β-葡萄糖苷酶的片段衍生调节剂

Eleni Makraki ,John F Darby ,Marta G Carneiro ,James D Firth ,Alex Heyam ,Eiso Ab ,Peter O'Brien ,Gregg Siegal ,Roderick E Hubbard

Exploring IDP-Ligand Interactions: tau K18 as A Test Case

探索 IDP-配体相互作用:以 tau K18 为例

Darius Vagrys, James Davidson, Ijen Chen, Roderick E Hubbard, Ben Davis

Fragment approaches in structure-based drug discovery

基于结构的药物发现中的片段方法

Roderick E Hubbard

Delineation of a unique protein-protein interaction site on the surface of the estrogen receptor

雌激素受体表面独特的蛋白质-蛋白质相互作用位点的描绘

Eric H Kong, Nina Heldring, Jan-Ake Gustafsson, Eckardt Treuter, Roderick E Hubbard, Ashley C W Pike