日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

HTRF-based identification of small molecules targeting SARS-CoV-2 E protein interaction with ZO-1 PDZ2

基于HTRF的靶向SARS-CoV-2 E蛋白与ZO-1 PDZ2相互作用的小分子鉴定

Alvarez, Flavio; Larrous, Florence; Mechaly, Ariel; Bardiaux, Benjamin; Goor, Quentin; Haouz, Ahmed; Séon-Méniel, Blandine; de Sousa, Rodolphe Alves; Bourg, Stéphane; Desmaële, Didier; Figadère, Bruno; Wolff, Nicolas; Munier-Lehmann, Hélène; Caillet-Saguy, Célia

Targeting Degradation of EGFR through the Allosteric Site Leads to Cancer Cell Detachment-Promoted Death

通过变构位点靶向降解 EGFR 可导致癌细胞脱离并死亡

Melkon Iradyan, Nina Iradyan, Philippe Hulin, Artur Hambardzumyan, Aram Gyulkhandanyan, Rodolphe Alves de Sousa, Assia Hessani, Christos Roussakis, Guillaume Bollot, Cyril Bauvais, Vehary Sakanyan

A Novel Polyaminocarboxylate Compound To Treat Murine Pulmonary Aspergillosis by Interfering with Zinc Metabolism

一种新型聚氨基羧酸酯化合物通过干扰锌代谢治疗小鼠肺曲霉病

Laskaris, Paris; Vicentefranqueira, Rocío; Helynck, Olivier; Jouvion, Grégory; Calera, José Antonio; du Merle, Laurence; Suzenet, Franck; Buron, Frédéric; de Sousa, Rodolphe Alves; Mansuy, Daniel; Cavaillon, Jean-Marc; Latgé, Jean-Paul; Munier-Lehmann, Hélène; Ibrahim-Granet, Oumaima

Activation of EGFR by small compounds through coupling the generation of hydrogen peroxide to stable dimerization of Cu/Zn SOD1

小分子化合物通过将过氧化氢的生成与 Cu/Zn SOD1 的稳定二聚化相结合来激活 EGFR

Vehary Sakanyan, Philippe Hulin, Rodolphe Alves de Sousa, Viviane A O Silva, Artur Hambardzumyan, Steven Nedellec, Christophe Tomasoni, Cédric Logé, Charles Pineau, Christos Roussakis, Fabrice Fleury, Isabelle Artaud