Glucosylpolyphenols as Inhibitors of Aβ-Induced Fyn Kinase Activation and Tau Phosphorylation: Synthesis, Membrane Permeability, and Exploratory Target Assessment within the Scope of Type 2 Diabetes and Alzheimer's Disease
葡萄糖多酚作为 Aβ 诱导的 Fyn 激酶活化和 Tau 磷酸化的抑制剂:合成、膜通透性和 2 型糖尿病和阿尔茨海默病范围内的探索性靶标评估
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.0c00841
Ana M de Matos, M Teresa Blázquez-Sánchez, Andreia Bento-Oliveira, Rodrigo F M de Almeida, Rafael Nunes, Pedro E M Lopes, Miguel Machuqueiro, Joana S Cristóvão, Cláudio M Gomes, Cleide S Souza, Imane G El Idrissi, Nicola A Colabufo, Ana Diniz, Filipa Marcelo, M Conceição Oliveira, Óscar López, José