日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Small molecule inhibition of the CBFβ/RUNX interaction decreases ovarian cancer growth and migration through alterations in genes related to epithelial-to-mesenchymal transition

小分子抑制 CBFβ/RUNX 相互作用可通过改变上皮-间质转化相关基因来降低卵巢癌的生长和迁移

Anne L Carlton, Anuradha Illendula, Yan Gao, Danielle C Llaneza, Adam Boulton, Anant Shah, Roger A Rajewski, Charles N Landen, David Wotton, John H Bushweller

A second-generation 2-Methoxyestradiol prodrug is effective against Barrett's adenocarcinoma in a mouse xenograft model

第二代 2-甲氧基雌二醇前药对小鼠异种移植模型中的巴雷特腺癌有效

Suman Kambhampati, Roger A Rajewski, Mehmet Tanol, Inamul Haque, Amlan Das, Snigdha Banerjee, Saheli Jha, Douglas Burns, Emma Borrego-Diaz, Peter J Van Veldhuizen, Sushanta K Banerjee

Development and characterization of a novel C-terminal inhibitor of Hsp90 in androgen dependent and independent prostate cancer cells

雄激素依赖性和非雄激素依赖性前列腺癌细胞中 Hsp90 新型 C 端抑制剂的开发和表征

Jeffery D Eskew, Takrima Sadikot, Pedro Morales, Alicia Duren, Irene Dunwiddie, Megan Swink, Xiaoying Zhang, Stacey Hembruff, Alison Donnelly, Roger A Rajewski, Brian S J Blagg, Jacob R Manjarrez, Robert L Matts, Jeffrey M Holzbeierlein, George A Vielhauer

Phase 0 clinical chemoprevention trial of the Akt inhibitor SR13668

Akt 抑制剂 SR13668 的 0 期临床化学预防试验

Joel M Reid, Chad A Walden, Rui Qin, Katie L Allen Ziegler, John L Haslam, Roger A Rajewski, Roger Warndahl, Cindy L Fitting, Daniel Boring, Eva Szabo, James Crowell, Marjorie Perloff, Ling Jong, Brent A Bauer, Sumithra J Mandrekar, Matthew M Ames, Paul J Limburg; Cancer Prevention Network