日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

TRPtracker: a community database for monitoring praziquantel sensitivity at TRPM(PZQ) variants

TRPtracker:一个用于监测TRPM(PZQ)变异株吡喹酮敏感性的社区数据库

Rohr, Claudia M; Park, Sang-Kyu; Aguiar-Martins, Kelsilandia; Anderson, Timothy J C; Berger, Duncan J; Berriman, Matthew; Buddenborg, Sarah K; Bustinduy, Amaya L; Chevalier, Frédéric D; Cotton, James A; Crellen, Thomas; Doyle, Stephen R; Emery, Aidan M; Kincaid Smith, Julien; Kinung'hi, Safari; Lamberton, Poppy H L; Le Clec'h, Winka; Ndombi, Eric; Pennance, Tom; Rowel, Candia; Summers, Shannan S; Tushabe, John Vianney; Walker, Martin; Webster, Bonnie L; Webster, Joanne P; Wilson, Shona; Marchant, Jonathan S

Meclonazepam sensitivity of parasitic flatworms correlates with TRPM(MCLZ) sensitivity to meclonazepam

寄生扁形动物对美氯硝西泮的敏感性与TRPM(MCLZ)对美氯硝西泮的敏感性相关

Rohr, Claudia M; McCusker, Paul; Kaethner, Marc; Armstrong, Rebecca; Robb, Emily; Park, Sang-Kyu; Sprague, Daniel J; Maule, Aaron G; Zamanian, Mostafa; Lundström-Stadelmann, Britta; Chan, John D; Marchant, Jonathan S

Target-Based Design of Praziquantel Analogs at Cestode TRPM(PZQ)

基于靶点的吡喹酮类似物设计(针对绦虫 TRPM(PZQ))

Sprague, Daniel J; Park, Sang-Kyu; Kaethner, Marc; Rohr, Claudia M; Ghobrial, Mina R; Barth, D Connor; Maillard, David; Spangenberg, Thomas; Lundström-Stadelmann, Britta; Marchant, Jonathan S

TRPtracker: a community database for monitoring praziquantel sensitivity at TRPM(PZQ) variants

TRPtracker:一个用于监测TRPM(PZQ)变异株吡喹酮敏感性的社区数据库

Rohr, Claudia M; Park, Sang-Kyu; Aguiar-Martins, Kelsilandia; Anderson, Timothy J C; Berger, Duncan J; Berriman, Matthew; Buddenborg, Sarah K; Bustinduy, Amaya L; Chevalier, Frédéric D; Cotton, James A; Crellen, Thomas; Doyle, Stephen R; Emery, Aidan M; Smith, Julien Kincaid; Kinung'hi, Safari; Lamberton, Poppy H L; Le Clec'h, Winka; Ndombi, Eric; Pennance, Tom; Rowel, Candia; Summers, Shannan S; Tushabe, John Vianney; Walker, Martin; Webster, Bonnie L; Webster, Joanne P; Wilson, Shona; Marchant, Jonathan S

Target-based discovery of a broad-spectrum flukicide.

基于靶点的广谱杀吸虫剂的发现

Sprague Daniel J, Park Sang-Kyu, Gramberg Svenja, Bauer Lisa, Rohr Claudia M, Chulkov Evgeny G, Smith Emery, Scampavia Louis, Spicer Timothy P, Haeberlein Simone, Marchant Jonathan S

The anthelmintic meclonazepam activates a schistosome transient receptor potential channel

驱虫药美氯硝西泮可激活血吸虫瞬时受体电位通道。

Park, Sang-Kyu; Sprague, Daniel J; Rohr, Claudia M; Chulkov, Evgeny G; Petrow, Ian; Kumar, Sushil; Marchant, Jonathan S

TRP drop, TRP drop: a steady patter of anti-schistosomal target illumination

TRP下降,TRP下降:抗血吸虫靶标照明的稳定模式

Sprague, Daniel J; Rohr, Claudia M; Marchant, Jonathan S

Natural variation in the binding pocket of a parasitic flatworm TRPM channel resolves the basis for praziquantel sensitivity.

寄生扁形动物 TRPM 通道结合口袋的自然变异揭示了吡喹酮敏感性的基础

Rohr Claudia M, Sprague Daniel J, Park Sang-Kyu, Malcolm Nicholas J, Marchant Jonathan S

The Anthelmintic Activity of Praziquantel Analogs Correlates with Structure-Activity Relationships at TRPM(PZQ) Orthologs

吡喹酮类似物的驱虫活性与TRPM(PZQ)同源物的构效关系相关

Sprague, Daniel J; Kaethner, Marc; Park, Sang-Kyu; Rohr, Claudia M; Harris, Jade L; Maillard, David; Spangenberg, Thomas; Lundström-Stadelmann, Britta; Marchant, Jonathan S

Praziquantel activates a native cation current in Schistosoma mansoni

吡喹酮激活曼氏血吸虫体内的固有阳离子电流

Chulkov, Evgeny G; Rohr, Claudia M; Marchant, Jonathan S