Preclinical profile of a potent gamma-secretase inhibitor targeting notch signaling with in vivo efficacy and pharmacodynamic properties
针对 Notch 信号的强效 γ-分泌酶抑制剂的临床前概况,具有体内功效和药效学特性
期刊:Cancer Research
影响因子:12.5
doi:10.1158/0008-5472.CAN-09-1843
Leopoldo Luistro, Wei He, Melissa Smith, Kathryn Packman, Maria Vilenchik, Daisy Carvajal, John Roberts, James Cai, Windy Berkofsky-Fessler, Holly Hilton, Michael Linn, Alexander Flohr, Roland Jakob-Røtne, Helmut Jacobsen, Kelli Glenn, David Heimbrook, John F Boylan