日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Ophiobolin A impacts mitochondrial redox biology in an epithelial-mesenchymal transition (EMT)-specific manner.

Ophiobolin A 以上皮-间质转化 (EMT) 特异性方式影响线粒体氧化还原生物学。

Parker Haleigh N, Tao Yongfeng, Tobin Jenna, Haberman Kayla L, Davis Samantha, York Emily, Martinez Alysia, Matsumoto Nobuyuki, Aroujo Jaquelin, Park Jun Hyoung, Zechmann Bernd, Kaipparettu Benny Abraham, Boari Angela, Sayes Christie M, Evidente Antonio, Kornienko Alexander, Cravatt Benjamin, Romo Daniel, Taube Joseph H

Gasdermin D Cleavage and Cytokine Release, Indicative of Pyroptotic Cell Death, Induced by Ophiobolin A in Breast Cancer Cell Lines.

Gasdermin D 裂解和细胞因子释放,表明 Ophiobolin A 在乳腺癌细胞系中诱导细胞焦亡。

Ranganathan Santhalakshmi, Ojo Tolulope, Subramanian Alagu, Tobin Jenna, Kornienko Alexander, Boari Angela, Evidente Antonio, Benton Mary Lauren, Romo Daniel, Taube Joseph H

Gigobolins A-C, New Ophiobolins with Anticancer Activity from the Phytopathogenic Fungus Drechslera gigantea

从植物病原真菌巨孢菌(Drechslera gigantea)中分离得到的具有抗癌活性的新型蛇形素类化合物Gigobolins AC

Carbone, Marianna; Jayamohan, Sridharan; Scott, Amelia; Boari, Angela; Rutledge, Ryan J; Cacciapuoti, Nadia; Gautam, Vamika; Aroujo, Jaquelin; Betancourt, Tania; Romo, Daniel; Sareddy, Gangadhara Reddy; Taube, Joseph H; Kornienko, Alexander; Evidente, Antonio; Ciavatta, Maria Letizia

Intramolecular epistasis correlates with divergence of specificity in promiscuous and bifunctional NSAR/OSBS enzymes.

分子内上位性与混杂型和双功能 NSAR/OSBS 酶的特异性差异相关

Truong Dat P, Dharmatti Roopa, Suriadinata Dylan, Huddleston Jamison, Skouby Rebecca, Owusu Addo Gladys, Zhu Mingzhao, Acharige Anjana Delpe, Sankari Bayana Reethu, Davila Cristian, Fults Susan C, Raushel Frank M, Hull Kenneth G, Romo Daniel, Glasner Margaret E

Derivatization of ophiobolin A and cytotoxicity toward breast and glioblastoma cancer stem cells: Varying the ketone and unsaturated aldehyde moieties

蛇毒素A的衍生化及其对乳腺癌和胶质母细胞瘤癌干细胞的细胞毒性:改变酮基和不饱和醛基

Aroujo, Jaquelin; Parker, Haleigh; Boari, Angela; Mason, Evan; Otakpor, Mackenzie U; Betancourt, Tania; Kornienko, Alexander; Ciavatta, Maria Letizia; Carbone, Marianna; Evidente, Antonio; Taube, Joseph H; Romo, Daniel

Dopamine-Derived Guanidine Alkaloids from a Didemnidae Tunicate: Isolation, Synthesis, and Biological Activities

从海鞘科海鞘中分离、合成并研究了多巴胺衍生的胍类生物碱的生物活性。

Sakai, Ryuichi; Matsumura, Ken; Uchimasu, Hajime; Miyako, Kei; Taniguchi, Tohru; Kovvuri, V Raghavendra Rao; Acharige, Anjana Delpe; Hull, Kenneth G; Romo, Daniel; Thaveepornkul, Lakkana; Chimnaronk, Sarin; Miyamoto, Hiroko; Takada, Ayato; Watari, Hiromi; Fujita, Masaki J; Sakaue, Jiro

Therapeutic vulnerabilities of cancer stem cells and effects of natural products

癌症干细胞的治疗弱点及天然产物的作用

Reisenauer, Keighley N; Aroujo, Jaquelin; Tao, Yongfeng; Ranganathan, Santhalakshmi; Romo, Daniel; Taube, Joseph H

Zinc-mediated carboxylations of allylic and propargylic halides in flow: synthesis of β-lactones via subsequent bromolactonization

流动条件下锌介导的烯丙基和炔丙基卤化物羧化反应:通过后续溴代内酯化反应合成β-内酯

Sutter, Patrick J; Kang, Guowei; Vellalath, Sreekumar; Romo, Daniel

Total Synthesis of (±)-N-Methyldibromoisophakellin and N-Methylugibohlin via Net [3+2] Cycloguanidinylations Employing 2-Amido-1,3-Diamino-Allyl Cations

利用 2-酰胺基-1,3-二氨基烯丙基阳离子,通过 [3+2] 环胍基化反应全合成 (±)-N-甲基二溴异叶绿素和 N-甲基乌吉布林。

Matsumoto, Nobuyuki; Hwang, Taehwan; Romo, Daniel

Enzymatic assembly of the salinosporamide γ-lactam-β-lactone anticancer warhead

盐霉素γ-内酰胺-β-内酯抗癌弹头的酶促组装

Bauman, Katherine D; Shende, Vikram V; Chen, Percival Yang-Ting; Trivella, Daniela B B; Gulder, Tobias A M; Vellalath, Sreekumar; Romo, Daniel; Moore, Bradley S