日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Systematic elucidation and pharmacological targeting of tumor-infiltrating regulatory T cell master regulators

系统阐明和药理学靶向肿瘤浸润调节性T细胞主调控因子

Aleksandar Obradovic ,Casey Ager ,Mikko Turunen ,Thomas Nirschl ,Mohsen Khosravi-Maharlooei ,Alina Iuga ,Christopher M Jackson ,Srinivasan Yegnasubramanian ,Lorenzo Tomassoni ,Ester Calvo Fernandez ,Patrick McCann ,Meri Rogava ,Angelo M DeMarzo ,Christina M Kochel ,Mohamad Allaf ,Trinity Bivalacqua ,Michael Lim ,Ronald Realubit ,Charles Karan ,Charles G Drake ,Andrea Califano

TOP2B Enzymatic Activity on Promoters and Introns Modulates Multiple Oncogenes in Human Gliomas

启动子和内含子上的 TOP2B 酶活性调节人类胶质瘤中的多种致癌基因

Edgar Gonzalez-Buendia #, Junfei Zhao #, Lu Wang, Subhas Mukherjee, Daniel Zhang, Víctor A Arrieta, Eric Feldstein, J Robert Kane, Seong Jae Kang, Catalina Lee-Chang, Aayushi Mahajan, Li Chen, Ronald Realubit, Charles Karan, Lisa Magnuson, Craig Horbinski, Stacy A Marshall, Jann N Sarkaria, Ahmed Mo

Systematic, network-based characterization of therapeutic target inhibitors

治疗靶点抑制剂的系统、基于网络的表征

Yao Shen, Mariano J Alvarez, Brygida Bisikirska, Alexander Lachmann, Ronald Realubit, Sergey Pampou, Jorida Coku, Charles Karan, Andrea Califano

A novel, rapid method to compare the therapeutic windows of oral anticoagulants using the Hill coefficient

一种使用希尔系数比较口服抗凝剂治疗窗口的新型快速方法

Jeremy B Chang, Kayla M Quinnies, Ronald Realubit, Charles Karan, Jacob H Rand, Nicholas P Tatonetti

Elucidating Compound Mechanism of Action by Network Perturbation Analysis

通过网络扰动分析阐明化合物的作用机制

Jung Hoon Woo, Yishai Shimoni, Wan Seok Yang, Prem Subramaniam, Archana Iyer, Paola Nicoletti, María Rodríguez Martínez, Gonzalo López, Michela Mattioli, Ronald Realubit, Charles Karan, Brent R Stockwell, Mukesh Bansal, Andrea Califano

Preclinical pharmacologic evaluation of pralatrexate and romidepsin confirms potent synergy of the combination in a murine model of human T-cell lymphoma

普拉曲沙和罗米地辛的临床前药理学评估证实了该组合在人类 T 细胞淋巴瘤小鼠模型中具有强大的协同作用

Salvia Jain, Xavier Jirau-Serrano, Kelly M Zullo, Luigi Scotto, Carmine F Palermo, Stephen A Sastra, Kenneth P Olive, Serge Cremers, Tiffany Thomas, Ying Wei, Yuan Zhang, Govind Bhagat, Jennifer E Amengual, Changchun Deng, Charles Karan, Ronald Realubit, Susan E Bates, Owen A O'Connor

Simulating henipavirus multicycle replication in a screening assay leads to identification of a promising candidate for therapy

在筛选试验中模拟亨尼巴病毒的多周期复制可确定有希望的治疗候选药物

Matteo Porotto, Gianmarco Orefice, Christine C Yokoyama, Bruce A Mungall, Ronald Realubit, Michael L Sganga, Mohamad Aljofan, Michael Whitt, Fraser Glickman, Anne Moscona