日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

4-(5-Chloro-3-(3,4,5-trimethoxybenzoyl)-1H-indol-1-yl)benzenesulfonamide: A Novel Polypharmacology Agent to Target Carbonic Anhydrase IX and XII With Improved Selectivity, Wnt/β-Catenin Signaling Pathway, and P-Glycoprotein

4-(5-氯-3-(3,4,5-三甲氧基苯甲酰基)-1H-吲哚-1-基)苯磺酰胺:一种新型多靶点药物,可选择性地靶向碳酸酐酶IX和XII、Wnt/β-catenin信号通路以及P-糖蛋白。

Puxeddu, Michela; Bordone, Rosa; Colla, Claudia; Rotili, Gabriele; Coluccia, Antonio; Sciò, Pietro; Cuřínová, Petra; Nocentini, Alessio; Supuran, Claudiu T; Filiberti, Serena; Turati, Marta; Ronca, Roberto; Kopecka, Joanna; Riganti, Chiara; Jimenez, Lucia; Link, Wolfgang; Bigogno, Chiara; Dondio, Giulio; Barba, Martina; Canettieri, Gianluca; Silvestri, Romano; La Regina, Giuseppe

An ureido-substituted benzenesulfonamide carbonic anhydrase inhibitor exerts a potent antitumor effect in vitro and in vivo

一种脲基取代的苯磺酰胺类碳酸酐酶抑制剂在体外和体内均表现出显著的抗肿瘤作用。

Gazzaroli, Giorgia; Tavani, Camilla; Filiberti, Serena; Massardi, Maria Luisa; Turati, Marta; Garattini, Giulia; Peat, Thomas S; Pieraccini, Giuseppe; Angeli, Andrea; Supuran, Claudiu T; Carta, Fabrizio; Giacomini, Arianna; Ronca, Roberto

A Glucosylated BODIPY Uses the GLUT Channel to Target Cancer Cells in In Vitro and In Vivo Models

糖基化BODIPY利用GLUT通道在体外和体内模型中靶向癌细胞

Turati, Marta; Biagiotti, Giacomo; Ravelli, Cosetta; Tobia, Chiara; Cardellini, Jacopo; Mignani, Luca; Tricomi, Jacopo; Berti, Debora; Cicchi, Stefano; Richichi, Barbara; Ronca, Roberto

Selective Inhibition of Carbonic Anhydrase IX and XII by Natural Coumarin Coladonin and Its Derivatives: Promising Antimelanoma and Antiglioblastoma Agents

天然香豆素可乐多宁及其衍生物对碳酸酐酶IX和XII的选择性抑制:有前景的抗黑色素瘤和抗胶质母细胞瘤药物

Mustafa, Muhamad; Baccari, Wiem; Nocentini, Alessio; Massardi, Maria Luisa; Smietana, Michael; Abbass, Eslam M; Saidi, Ilyes; Znati, Mansour; Ben Jannet, Hichem; Ronca, Roberto; Supuran, Claudiu T; Winum, Jean-Yves

Pegylation approach applied to erlotinib-carbonic anhydrase inhibitors hybrids towards anticancer agents

聚乙二醇化方法应用于厄洛替尼-碳酸酐酶抑制剂杂合物,以开发抗癌药物

Filiberti, Serena; Renzi, Gioele; Carta, Fabrizio; Fantacuzzi, Marialuigia; D'Agostino, Ilaria; Benito, German; Angeli, Andrea; Massardi, Maria Luisa; Simsek, Rahime; Capasso, Clemente; Carradori, Simone; Ronca, Roberto; Supuran, Claudiu T

Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors

新型2,4-二氯-5-氨磺酰基苯甲酸肟酯:作为潜在的人类碳酸酐酶抑制剂的初步研究

Kilbile, Jaydeo T; Sapkal, Suryakant B; Renzi, Gioele; D'Agostino, Ilaria; Cutarella, Luigi; Mori, Mattia; De Filippis, Barbara; Islam, Imadul; Massardi, Maria Luisa; Somenza, Elena; Ronca, Roberto; Tamboli, Yasinalli; Carta, Fabrizio; Supuran, Claudiu T

Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity

苯磺酰胺修饰的二氢嘧啶(硫)酮:碳酸酐酶活性分析和抗增殖活性

Aslan, Hakan; Renzi, Gioele; Angeli, Andrea; D'Agostino, Ilaria; Ronca, Roberto; Massardi, Maria Luisa; Tavani, Camilla; Carradori, Simone; Ferraroni, Marta; Governa, Paolo; Manetti, Fabrizio; Carta, Fabrizio; Supuran, Claudiu T

Molecular Profiling of Lymphatic Endothelial Cell Activation In Vitro

体外淋巴内皮细胞活化的分子谱分析

Turati, Marta; Mattei, Gianluca; Boaretto, Alessia; Magi, Alberto; Calvani, Maura; Ronca, Roberto

The natural FGF-trap long pentraxin 3 inhibits lymphangiogenesis and lymphatic dissemination

天然FGF陷阱长链五聚蛋白3抑制淋巴管生成和淋巴扩散

Turati, Marta; Giacomini, Arianna; Rezzola, Sara; Maccarinelli, Federica; Gazzaroli, Giorgia; Valentino, Sonia; Bottazzi, Barbara; Presta, Marco; Ronca, Roberto

The lymphatic vasculature: An active and dynamic player in cancer progression

淋巴管系统:癌症进展中活跃且动态的角色

Rezzola, Sara; Sigmund, Elena C; Halin, Cornelia; Ronca, Roberto