日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of the SARS-CoV-2 Papain-Like Protease Inhibitor MR1-114: From Structure-Based Design to In Vivo Antiviral Efficacy

SARS-CoV-2木瓜蛋白酶样蛋白酶抑制剂MR1-114的发现:从基于结构的药物设计到体内抗病毒功效

Gannarapu, Malla Reddy; Indukuri, Divakar; Holberg, Cameron; Ratia, Kiira; Ramos, Omar Lozano; Cardoza, Savio; Velma, Ganga Reddy; Musku, Soumya Reddy; Qi, Zuohuang; Slilaty, Steve; Li, Zuomei; Rong, Lijun; Thatcher, Gregory R J; Xiong, Rui

Selective capture and digital counting of intact HIV pseudovirus using designer DNA nets, tethered motion, and photonic resonator interferometric scattering microscopy

利用人工设计的DNA网、系绳运动和光子谐振器干涉散射显微镜选择性捕获和数字化计数完整的HIV假病毒

Tibbs, Joseph; Umrao, Saurabh; Song, Tingjie; Anirudhan, Varada; Shepherd, Skye; Wolhaupter, Katy; Zheng, Mengxi; Wiggins, Sydney; Rong, Lijun; Hisey, Colin L; Demirci, Utkan; Wang, Xing; Cunningham, Brian T

Effect of pH on small-molecule inhibitor binding to influenza virus hemagglutinin

pH值对小分子抑制剂与流感病毒血凝素结合的影响

Anirudhan, Varada; Gaisina, Irina; Shimon, Amir; Lee, Hyun; Alqarni, Saad; Manicassamy, Balaji; Moore, Terry W; Xu, Kai; Caffrey, Michael; Rong, Lijun

Cryo-EM structures of Nipah virus polymerase complex reveal highly varied interactions between L and P proteins among paramyxoviruses.

尼帕病毒聚合酶复合物的冷冻电镜结构揭示了副黏病毒中 L 蛋白和 P 蛋白之间高度多样化的相互作用

Xue Lu, Chang Tiancai, Gui Jiacheng, Li Zimu, Zhao Heyu, Zou Binqian, Lu Junnan, Li Mei, Wen Xin, Gao Shenghua, Zhan Peng, Rong Lijun, Feng Liqiang, Gong Peng, He Jun, Chen Xinwen, Xiong Xiaoli

Engineering Two-Dimensional Nanobody-Origami Architectures for Enhanced Antiviral Activity

构建二维纳米抗体折纸结构以增强抗病毒活性

Song, Tingjie; Galván Achi, Jazmin; Anirudhan, Varada; Gandavadi, Dhanush; Le, Linh T P; Hammound, Kadmos C; Morshed, Mehzabin; Wang, Xiaojing; Rong, Lijun; Wang, Xing

Mechanistic insights into the small-molecule inhibition of influenza A virus entry.

对小分子抑制甲型流感病毒入侵的机制研究。

Xu Yan, Anirudhan Varada, Gaisina Irina N, Du Haijuan, Alqarni Saad, Moore Terry W, Caffrey Michael, Manicassamy Balaji, Zhou Tongqing, Rong Lijun, Xu Kai

Guardians at the Gate: Optimization of Small Molecule Entry Inhibitors of Ebola and Marburg Viruses.

守门人:埃博拉病毒和马尔堡病毒小分子进入抑制剂的优化

Argade Malaika D, Achi Jazmin Galván, Bott Ryan, Morsheimer Kimberly M, Owen Callum D, Zielinski Christian A, Gaisin Arsen M, Alvarez Mario, Moore Terry W, Bu Fan, Li Fang, Cameron Michael, Anantpadma Manu, Davey Robert A, Peet Norton P, Rong Lijun, Gaisina Irina N

Selective Degradation and Inhibition of SARS-CoV-2 3CL(pro) by MMP14 Reveals a Novel Strategy for COVID-19 Therapeutics

MMP14对SARS-CoV-2 3CL(pro)的选择性降解和抑制揭示了一种治疗COVID-19的新策略

Lee, Hyun; Hwang, Yunjeong; Mulder, Elizabeth J; Song, Yuri; Choi, Calista; Rong, Lijun; Azar, Dimitri T; Han, Kyu-Yeon

Inhibition of Influenza Entry by Organosilicon Compounds

有机硅化合物对流感病毒入侵的抑制作用

Antanasijevic, Aleksandar; Haferman, Nicholas J; Shimon, Amir; Tundup, Smanla; Anirudhan, Varada; Rong, Lijun; Manicassamy, Balaji; Wardrop, Duncan; Caffrey, Michael

Small molecule drug discovery for Ebola virus disease

埃博拉病毒病的小分子药物研发

Durante, Destiny; Murugesh, Venkatesh; Kalanquin, Tyler; Gaisina, Irina N; Rong, Lijun; Moore, Terry W