日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacological targeting of RIG-I can selectively activate the integrated stress response

通过药物靶向RIG-I可以选择性地激活整合应激反应。

Cuoco, Caroline A; Ren, Wen; Baron, Kelsey R; Gologo, Sakina; Perea, Valerie; Mathur, Prakhyat; Bora, Prerona; Ta, Amina; Chu, Alan; Aldakhlallah, Rama; Rhoades, Derek; Cole, Christian M; Tan, Ee Phie; Hou, William C; Yoon, Leonard; Guo, Xiaoyan; Rosarda, Jessica D; Baran, Phil S; Kampmann, Martin; Tillery, Lakeisha; Johnson, Kristen A; Powers, Evan T; Wiseman, R Luke; Kelly, Jeffery W

Identification of a Selective Pharmacologic IRE1/XBP1s Activator with Enhanced Tissue Exposure.

鉴定一种具有增强组织暴露的选择性药理学IRE1/XBP1s激活剂。

Sun Jie, Lee Kyunga, Kutseikin Sergei, Guerrero Adrian, Rius Bibiana, Madhavan Aparajita, Buasakdi Chavin, Cheong Ka-Neng, Chatterjee Priyadarshini, Rosen Dorian A, Yoon Leonard, Ardejani Maziar S, Mendoza Alejandra, Rosarda Jessica D, Saez Enrique, Kelly Jeffery W, Wiseman R Luke

Covalent Targeting As a Common Mechanism for Inhibiting NLRP3 Inflammasome Assembly

共价靶向作为抑制 NLRP3 炎症小体组装的常见机制

Caroline Stanton, Jie Sun, Kayla Nutsch, Jessica D Rosarda, Thu Nguyen, Chloris Li-Ma, Evert Njomen, Bruno Melillo, Sergei Kutseikin, Enrique Saez, Benjamin F Cravatt, John R Teijaro, R Luke Wiseman, Michael J Bollong

Metabolically activated proteostasis regulators that protect against erastin-induced ferroptosis

代谢激活的蛋白质稳态调节因子可防止erastin诱导的铁死亡

Kline, Gabriel M; Madrazo, Nicole; Cole, Christian M; Pannikkat, Meera; Bollong, Michael J; Rosarda, Jessica D; Kelly, Jeffery W; Wiseman, R Luke

Mapping stress-responsive signaling pathways induced by mitochondrial proteostasis perturbations

绘制线粒体蛋白质稳态扰动诱导的应激反应信号通路图

Madrazo, Nicole; Khattar, Zinia; Powers, Evan T; Rosarda, Jessica D; Wiseman, R Luke

Pharmacologic Targeting of PDIA1 Inhibits NLRP3 Inflammasome Assembly and Activation.

PDIA1 的药理学靶向作用可抑制 NLRP3 炎症小体的组装和激活

Rosarda Jessica D, Stanton Caroline R, Chen Emily B, Bollong Michael J, Wiseman R Luke

Mapping Stress-Responsive Signaling Pathways Induced by Mitochondrial Proteostasis Perturbations

绘制线粒体蛋白质稳态扰动诱导的应激反应信号通路图谱

Madrazo, Nicole; Khattar, Zinia; Powers, Evan T; Rosarda, Jessica D; Wiseman, R Luke

Imbalanced unfolded protein response signaling contributes to 1-deoxysphingolipid retinal toxicity

不平衡的未折叠蛋白反应信号导致1-脱氧鞘脂视网膜毒性

Jessica D Rosarda, Sarah Giles, Sarah Harkins-Perry, Elizabeth A Mills, Martin Friedlander, R Luke Wiseman, Kevin T Eade

Pharmacologic activation of a compensatory integrated stress response kinase promotes mitochondrial remodeling in PERK-deficient cells

药理学激活补偿性整合应激反应激酶可促进PERK缺陷细胞的线粒体重塑。

Valerie Perea ,Kelsey R Baron ,Vivian Dolina ,Giovanni Aviles ,Grace Kim ,Jessica D Rosarda ,Xiaoyan Guo ,Martin Kampmann ,R Luke Wiseman

Covalent targeting as a common mechanism for inhibiting NLRP3 inflammasome assembly

共价靶向是抑制 NLRP3 炎症小体组装的常见机制

Caroline Stanton, Jie Sun, Kayla Nutsch, Jessica D Rosarda, Thu Nguyen, Chloris Li-Ma, Sergei Kutseikin, Enrique Saez, John R Teijaro, R Luke Wiseman, Michael J Bollong