M4205 (IDRX-42) Is a Highly Selective and Potent Inhibitor of Relevant Oncogenic Driver and Resistance Variants of KIT in Cancer.
M4205 (IDRX-42) 是一种对癌症中 KIT 相关致癌驱动因子和耐药变体具有高度选择性和强效抑制作用的抑制剂
期刊:Molecular Cancer Therapeutics
影响因子:5.5
doi:10.1158/1535-7163.MCT-24-0699
Esdar Christina, Linde Nina, Blum Andreas, Schieferstein Hanno, Drechsler Christine, Sherbetjian Eva, Petersson Carl, Ross Edith, Leuthner Birgitta, Grädler Ulrich, Dorsch Dieter, Blaukat Andree