Design, Synthesis, Biological Evaluation, and Computational Studies of Novel Ureidopropanamides as Formyl Peptide Receptor 2 (FPR2) Agonists to Target the Resolution of Inflammation in Central Nervous System Disorders
新型脲基丙酰胺作为甲酰肽受体 2 (FPR2) 激动剂的设计、合成、生物学评价和计算研究,旨在缓解中枢神经系统疾病的炎症
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.1c02203
Margherita Mastromarino, Maria Favia, Igor A Schepetkin, Lylia N Kirpotina, Ewa Trojan, Mauro Niso, Antonio Carrieri, Monika Leśkiewicz, Magdalena Regulska, Massimiliano Darida, Francesco Rossignolo, Stefano Fontana, Mark T Quinn, Agnieszka Basta-Kaim, Marcello Leopoldo, Enza Lacivita