日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

G(z) and β-arrestin 1 signaling in the μ-opioid receptor

μ-阿片受体中的G(z)和β-arrestin 1信号传导

Cheng, Zhi; Roth, Bryan L

Structure-based design of an opioid receptor modulator for enhanced morphine analgesia

基于结构的阿片受体调节剂设计及其在增强吗啡镇痛中的应用

Wang, Yue; Luo, Ping; Xu, Haiyan; Zhan, Li; Sakamoto, Kensuke; Li, Mingyu; Wang, Jing; Huang, Xi-Ping; Zhou, Jianhui; Liu, Tao; Suo, Yanrui; Fan, Wenjia; He, Xinheng; Xu, Youwei; Cai, Yongjie; Wang, Chao; Zhao, Yuxi; Dai, Antao; Lai, Yali; Yuan, Qingning; Hu, Wen; Wu, Kai; Yang, Dehua; Cheng, Xi; Lu, Xiaojie; Krumm, Brian; Kenakin, Terry; Zhang, Jian; Roth, Bryan L; Gao, Zhaobing; Xu, H Eric; Zhuang, Youwen

Structural insights into coffee bitter taste perception by TAS2R43 receptor

TAS2R43受体对咖啡苦味感知的结构性见解

Kim, Yoojoong; Gumpper, Ryan H; Zhuang, Yuxuan; Dror, Ron O; Roth, Bryan L

Large Library Docking for Polypharmacology

用于多药理学的大型库对接

Wu, Yujin; Vigneron, Seth; Braz, Joao; Srinivasan, Karthik; Fink, Elissa A; Huang, Xi-Ping; Xu, Xinyu; Huebner, Harald; Kim, Joseph Y; Wang, Jing; Pfeiffer, Tara; Sakamoto, Kensuke; Radchenko, Dmytro S; Rodriguiz, Ramona M; Moroz, Yurii S; Irwin, John J; Gmeiner, Peter; Billesboelle, Christian; Roth, Bryan L; Basbaum, Allan I; Manglik, Aashish; Wetsel, William C; Shoichet, Brian K

Cryo-EM Structures of Brain-Derived G Protein-Coupled Receptors: The First Direct Visualization from Mammalian Brain Tissue

脑源性G蛋白偶联受体的冷冻电镜结构:首次从哺乳动物脑组织中直接观察

Wright, Nicholas J; Chiu, Yi-Ting; Sakamoto, Kensuke; Kocak, D Dewran; Fordyce, Blake A; Hua, Kunjie; Huang, Karen Lu; Scherrer, Grégory; Lyons, Scott P; Roth, Bryan L

Xylazine's κ opioid agonist activity is not shared with other FDA-approved α(2)-adrenergic agonists

赛拉嗪的κ阿片受体激动剂活性与其他FDA批准的α(2)-肾上腺素能激动剂不同。

Huang, Xi-Ping; Krumm, Brian E; Bedard, Madigan L; McElligott, Zoe A; Roth, Bryan L

The selectivity implications of docking libraries with greater and lesser similarities to bio-like molecules

对接库与生物分子相似度高低的影响

Hall, Brendan W; Sakamoto, Kensuke; Huang, Xi-Ping; Irwin, John J; Shoichet, Brian K; Roth, Bryan L

Chemogenetics for sensing antigens

化学遗传学在抗原检测中的应用

Fordyce, Blake A; Roth, Bryan L

Orchestrating NTSR1 signaling from the interface

从接口协调 NTSR1 信号

Huang, Xianglin; Krumm, Brian E; Roth, Bryan L

The structural diversity of psychedelic drug actions revealed

迷幻药作用的结构多样性揭示

Gumpper, Ryan H; Jain, Manish K; Kim, Kuglae; Sun, Renhong; Sun, Ning; Xu, Zhongli; DiBerto, Jeffrey F; Krumm, Brian E; Kapolka, Nicholas J; Kaniskan, H Ümit; Nichols, David E; Jin, Jian; Fay, Jonathan F; Roth, Bryan L