日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of antibody-drug conjugate payloads that are substrates of ATP-binding cassette drug efflux transporters

鉴定抗体药物偶联物有效载荷,这些有效载荷是ATP结合盒药物外排转运体的底物

Roth, Jacob S; Guo, Hui; Chen, Lu; Shen, Min; Gbadegesin, Omotola; Robey, Robert W; Gottesman, Michael M; Hall, Matthew D

Identification of antibody-drug conjugate payloads which are substrates of ATP-binding cassette drug efflux transporters

鉴定抗体药物偶联物有效载荷,这些有效载荷是ATP结合盒药物外排转运体的底物

Roth, Jacob S; Guo, Hui; Chen, Lu; Shen, Min; Gbadegesin, Omotola; Robey, Robert W; Gottesman, Michael M; Hall, Matthew D

Loss of CARM1 alters the developmental programming of Glioma stem-like cells and creates a druggable NGFR/NTRK dependency.

CARM1 的缺失会改变胶质瘤干细胞样细胞的发育程序,并产生可药物靶向的 NGFR/NTRK 依赖性

Young Dejauwne L, Aguilan Jennifer, Cutler Ronald, Stransky Stephanie, DeAngelo Joseph D, Roth Jacob S, Malachowska Beata, Vercellino Justin, Bell Brett I, Shechter David, Tofilon Philip J, Phillips Richard E, Guha Chandan, Sidoli Simone

PRMT5 activity sustains histone production to maintain genome integrity.

PRMT5活性维持组蛋白的合成,从而保持基因组的完整性

Roth Jacob S, DeAngelo Joseph D, Young Dejauwne L, Maron Maxim I, Saha Ankita, Pinto Hugo, Gupta Varun, Jacobs Noah, Hegde Subray, Aguilan Jennifer T, Basken Joel, Azofeifa Joey, Query Charles C, Sidoli Simone, Skoultchi Arthur I, Shechter David

Remdesivir: A Review of Its Discovery and Development Leading to Emergency Use Authorization for Treatment of COVID-19

瑞德西韦:回顾其发现和研发历程,直至获得紧急使用授权用于治疗新冠肺炎

Eastman, Richard T; Roth, Jacob S; Brimacombe, Kyle R; Simeonov, Anton; Shen, Min; Patnaik, Samarjit; Hall, Matthew D

Correction to Remdesivir: A Review of Its Discovery and Development Leading to Human Clinical Trials for Treatment of COVID-19

关于瑞德西韦的更正:回顾其发现和研发历程,直至开展治疗新冠肺炎的人体临床试验

Eastman, Richard T; Roth, Jacob S; Brimacombe, Kyle R; Simeonov, Anton; Shen, Min; Patnaik, Samarjit; Hall, Matthew D

Keeping It Clean: The Cell Culture Quality Control Experience at the National Center for Advancing Translational Sciences

保持清洁:美国国家转化科学促进中心细胞培养质量控制经验

Roth, Jacob S; Lee, Tobie D; Cheff, Dorian M; Gosztyla, Maya L; Asawa, Rosita R; Danchik, Carina; Michael, Sam; Simeonov, Anton; Klumpp-Thomas, Carleen; Wilson, Kelli M; Hall, Matthew D

Canvass: A Crowd-Sourced, Natural-Product Screening Library for Exploring Biological Space

Canvass:一个用于探索生物空间的众包天然产物筛选库

Kearney, Sara E; Zahoránszky-Kőhalmi, Gergely; Brimacombe, Kyle R; Henderson, Mark J; Lynch, Caitlin; Zhao, Tongan; Wan, Kanny K; Itkin, Zina; Dillon, Christopher; Shen, Min; Cheff, Dorian M; Lee, Tobie D; Bougie, Danielle; Cheng, Ken; Coussens, Nathan P; Dorjsuren, Dorjbal; Eastman, Richard T; Huang, Ruili; Iannotti, Michael J; Karavadhi, Surendra; Klumpp-Thomas, Carleen; Roth, Jacob S; Sakamuru, Srilatha; Sun, Wei; Titus, Steven A; Yasgar, Adam; Zhang, Ya-Qin; Zhao, Jinghua; Andrade, Rodrigo B; Brown, M Kevin; Burns, Noah Z; Cha, Jin K; Mevers, Emily E; Clardy, Jon; Clement, Jason A; Crooks, Peter A; Cuny, Gregory D; Ganor, Jake; Moreno, Jesus; Morrill, Lucas A; Picazo, Elias; Susick, Robert B; Garg, Neil K; Goess, Brian C; Grossman, Robert B; Hughes, Chambers C; Johnston, Jeffrey N; Joullie, Madeleine M; Kinghorn, A Douglas; Kingston, David G I; Krische, Michael J; Kwon, Ohyun; Maimone, Thomas J; Majumdar, Susruta; Maloney, Katherine N; Mohamed, Enas; Murphy, Brian T; Nagorny, Pavel; Olson, David E; Overman, Larry E; Brown, Lauren E; Snyder, John K; Porco, John A Jr; Rivas, Fatima; Ross, Samir A; Sarpong, Richmond; Sharma, Indrajeet; Shaw, Jared T; Xu, Zhengren; Shen, Ben; Shi, Wei; Stephenson, Corey R J; Verano, Alyssa L; Tan, Derek S; Tang, Yi; Taylor, Richard E; Thomson, Regan J; Vosburg, David A; Wu, Jimmy; Wuest, William M; Zakarian, Armen; Zhang, Yufeng; Ren, Tianjing; Zuo, Zhong; Inglese, James; Michael, Sam; Simeonov, Anton; Zheng, Wei; Shinn, Paul; Jadhav, Ajit; Boxer, Matthew B; Hall, Matthew D; Xia, Menghang; Guha, Rajarshi; Rohde, Jason M