日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Phenomics-Based Discovery of Novel Orthosteric Choline Kinase Inhibitors

基于表型组学的新型正构胆碱激酶抑制剂的发现

Bauer, Ludwig G; Ward, Jennifer A; Díaz-Sáez, Laura; Sundström, Yvonne; Tolvanen, Tuomas; Alarcón Barrera, Juan Carlos; Kostidis, Sarantos; Rogers, Catherine M; Panagakou, Ioanna; Singh, Usha; Rothweiler, Elisabeth M; Gonzalez Orta, Alejandro; Kaniskan, H Ümit; Hu, Jianping; Jin, Jian; Sievers, Sonja; Waldmann, Herbert; Giera, Martin; Sundström, Michael; Berg, Louise; Huber, Kilian V M

A BRET biosensor for measuring uncompetitive engagement of PRMT5 complexes in cells.

一种用于测量细胞中 PRMT5 复合物非竞争性结合的 BRET 生物传感器。

Rothweiler Elisabeth M, Michaud Ani, Stefaniak Jakub, Singh Usha, Mikulsky Brynwood B, Vasta James D, Beck Michael T, Wilkinson Jennifer, Ward Jennifer A, Rogers Catherine M, Balıkçı Esra, Tranberg-Jensen Jeppe, Hansen Jesper S, Loppnau Peter, Whitty Adrian, Brennan Paul E, Tonge Peter J, Robers Matthew B, Huber Kilian V M

Covalent Inhibitors of KEAP1 with Exquisite Selectivity.

具有极高选择性的KEAP1共价抑制剂

Fejes Imre, Markacz Piroska, Tatai Janos, Rudas Monika, Dunkel Petra, Gyuris Mario, Nyerges Miklos, Provost Nicolas, Duvivier Valérie, Delerive Philippe, Martiny Virginie, Bristiel Alexandra, Vidal Brice, Richardson William, Rothweiler Elisabeth M, Tranberg-Jensen Jeppe, Manning Charlotte E, Sweeney Melissa N, Chalk Rod, Huber Kilian V M, Bullock Alex N, Herner Andras, Seedorf Klaus, Vinson Cedric, Weber Csaba, Kotschy Andras