The novel chemical entity YTR107 inhibits recruitment of nucleophosmin to sites of DNA damage, suppressing repair of DNA double-strand breaks and enhancing radiosensitization
新型化学实体 YTR107 可抑制核磷蛋白募集到 DNA 损伤位点,抑制 DNA 双链断裂修复并增强放射增敏作用
期刊:Clinical Cancer Research
影响因子:10
doi:10.1158/1078-0432.CCR-11-1054
Konjeti R Sekhar, Yerramreddy Thirupathi Reddy, Penthala Narsimha Reddy, Peter A Crooks, Amudhan Venkateswaran, William Hayes McDonald, Ling Geng, Soumya Sasi, Robert P Van Der Waal, Joseph L Roti Roti, Kenneth J Salleng, Girish Rachakonda, Michael L Freeman