日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

PROTAC-mediated degradation of Bcl-xL potentiates target therapy in preclinical melanoma models

PROTAC介导的Bcl-xL降解可增强黑色素瘤临床前模型中的靶向治疗效果

Valentini, Elisabetta; Gentile, Giulia; Di Martile, Marta; D'Aguanno, Simona; Brignone, Matteo; Di Stefano, Adriana Maria; Di Caprio, Marica; Melucci, Elisa; Botti, Claudio; Pelle, Fabio; Ortolano, Arianna; Fattore, Luigi; Mancini, Rita; Ciliberto, Gennaro; Rotili, Dante; Del Bufalo, Donatella

Dynamic epigenetic regulation of BCLAF1 splicing in acute myeloid leukemia

急性髓系白血病中BCLAF1剪接的动态表观遗传调控

Sgueglia, Giulia; Massaro, Crescenzo; Muro, Annamaria; Lettiero, Ida; D'Agostino, Erika; Favale, Gregorio; Simonelli, Nicla; Del Gaudio, Nunzio; Carafa, Vincenzo; De Marchi, Tommaso; Rotili, Dante; Valente, Sergio; Mai, Antonello; Sbardella, Gianluca; De Simone, Mariacarla; Altucci, Lucia; Dell'Aversana, Carmela

The ATC12 small molecule inhibits the Aurora-A/TPX2 interaction and impairs the proliferation of breast cancer cells

ATC12小分子抑制Aurora-A/TPX2相互作用,从而抑制乳腺癌细胞增殖。

Boi, Dalila; Fianco, Giulia; Polverino, Federica; Fiorentino, Francesco; Mastrangelo, Anna; Rossi, Simone; Rubini, Elisabetta; Rosignoli, Serena; Troilo, Francesca; Antonelli, Maria Rosaria; Tarquini, Dalila; Cervoni, Laura; Rinaldo, Serena; Tramonti, Angela; Scarpone, Eleonora Kristina; Naro, Chiara; Sette, Claudio; Stagni, Venturina; Colotti, Gianni; Rotili, Dante; Paiardini, Alessandro; Guarguaglini, Giulia; Asteriti, Italia Anna

4-(5-Chloro-3-(3,4,5-trimethoxybenzoyl)-1H-indol-1-yl)benzenesulfonamide: A Novel Polypharmacology Agent to Target Carbonic Anhydrase IX and XII With Improved Selectivity, Wnt/β-Catenin Signaling Pathway, and P-Glycoprotein

4-(5-氯-3-(3,4,5-三甲氧基苯甲酰基)-1H-吲哚-1-基)苯磺酰胺:一种新型多靶点药物,可选择性地靶向碳酸酐酶IX和XII、Wnt/β-catenin信号通路以及P-糖蛋白。

Puxeddu, Michela; Bordone, Rosa; Colla, Claudia; Rotili, Gabriele; Coluccia, Antonio; Sciò, Pietro; Cuřínová, Petra; Nocentini, Alessio; Supuran, Claudiu T; Filiberti, Serena; Turati, Marta; Ronca, Roberto; Kopecka, Joanna; Riganti, Chiara; Jimenez, Lucia; Link, Wolfgang; Bigogno, Chiara; Dondio, Giulio; Barba, Martina; Canettieri, Gianluca; Silvestri, Romano; La Regina, Giuseppe

Structural snapshots of Pseudomonas aeruginosa LptB(2)FG and LptB(2)FGC reveal insights into lipopolysaccharide recognition and transport.

铜绿假单胞菌 LptB(2)FG 和 LptB(2)FGC 的结构快照揭示了脂多糖识别和运输的见解。

Fiorentino Francesco, Cervoni Matteo, Wang Yi, Urner Leonhard H, Sauer Joshua B, Tran Anh, Corey Robin A, Rotili Dante, Mai Antonello, Stansfeld Phillip J, Imperi Francesco, Yu Edward W, Su Chih-Chia, Robinson Carol V, Bolla Jani R

Distinct viral reservoirs and immune signatures in individuals on long-term antiretroviral therapy with perinatally acquired HIV-1

接受长期抗逆转录病毒治疗的围产期感染 HIV-1 的个体中存在独特的病毒库和免疫特征

Benjamin Bone,Nicola Cotugno,Chiara Pighi,Arianna Rotili,Seohyun Hong,Leah Carrere,Elena Morrocchi,Giuseppe Rubens Pascucci,Ce Gao,Nicole Colantoni,Weiwei Sun,Giovanna Leone,David R Collins,Mpho J Olatotse,Giovanna Del Principe,Toong Seng Tan,Melanie Lancien,Alessia Neri,Libera Sessa,Giulio Olivieri,Kailey Shapiro,Isabelle Roseto,Catherine Koofhethile,Elena Emili,Stefania Bernardi,Ann Chahroudi,Paolo Rossi,Bruce D Walker,Xu G Yu,Mathias Lichterfeld,Paolo Palma

Distinct viral reservoirs and immune signatures in individuals on long-term antiretroviral therapy with perinatally acquired HIV-1

接受长期抗逆转录病毒治疗的围产期感染 HIV-1 的个体中存在独特的病毒库和免疫特征

Benjamin Bone ,Nicola Cotugno ,Chiara Pighi ,Arianna Rotili ,Seohyun Hong ,Leah Carrere ,Elena Morrocchi ,Giuseppe Rubens Pascucci ,Ce Gao ,Nicole Colantoni ,Weiwei Sun ,Giovanna Leone ,David R Collins ,Mpho J Olatotse ,Giovanna Del Principe ,Toong Seng Tan ,Melanie Lancien ,Alessia Neri ,Libera Sessa ,Giulio Olivieri ,Kailey Shapiro ,Isabelle Roseto ,Catherine Koofhethile ,Elena Emili ,Stefania Bernardi ,Ann Chahroudi ,Paolo Rossi ,Bruce D Walker ,Xu G Yu ,Mathias Lichterfeld ,Paolo Palma

Activation and inhibition of sirtuins: From bench to bedside

sirtuins 的激活和抑制:从实验室到临床

Fiorentino, Francesco; Fabbrizi, Emanuele; Mai, Antonello; Rotili, Dante

An Amazing 30-Year Journey around the DABO Family: A Medicinal Chemistry Lesson on a Versatile Class of Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors

DABO家族30年奇妙历程:一堂关于多功能非核苷类HIV-1逆转录酶抑制剂的药物化学课

Fabbrizi, Emanuele; Chernyshov, Vladimir V; Fiorentino, Francesco; Sbardella, Gianluca; Ragno, Rino; Nawrozkij, Maxim; Ivanov, Roman; Rotili, Dante; Mai, Antonello

A Combined SIRT5 Activation and SIRT3 Inhibition Prevents Breast Cancer Spheroids Growth by Reducing HIF-1α and Mitophagy

SIRT5激活和SIRT3抑制联合作用可通过减少HIF-1α和线粒体自噬来阻止乳腺癌球体的生长

Barreca, Federica; Aventaggiato, Michele; Cristina, Mario; Sansone, Luigi; Belli, Manuel; Lista, Maria Beatrice; Francisci, Gaia; Valente, Sergio; Rotili, Dante; Mai, Antonello; Russo, Matteo Antonio; Tafani, Marco