日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

PROTAC-mediated degradation of Bcl-xL potentiates target therapy in preclinical melanoma models

PROTAC介导的Bcl-xL降解可增强黑色素瘤临床前模型中的靶向治疗效果

Valentini, Elisabetta; Gentile, Giulia; Di Martile, Marta; D'Aguanno, Simona; Brignone, Matteo; Di Stefano, Adriana Maria; Di Caprio, Marica; Melucci, Elisa; Botti, Claudio; Pelle, Fabio; Ortolano, Arianna; Fattore, Luigi; Mancini, Rita; Ciliberto, Gennaro; Rotili, Dante; Del Bufalo, Donatella

Dynamic epigenetic regulation of BCLAF1 splicing in acute myeloid leukemia

急性髓系白血病中BCLAF1剪接的动态表观遗传调控

Sgueglia, Giulia; Massaro, Crescenzo; Muro, Annamaria; Lettiero, Ida; D'Agostino, Erika; Favale, Gregorio; Simonelli, Nicla; Del Gaudio, Nunzio; Carafa, Vincenzo; De Marchi, Tommaso; Rotili, Dante; Valente, Sergio; Mai, Antonello; Sbardella, Gianluca; De Simone, Mariacarla; Altucci, Lucia; Dell'Aversana, Carmela

The ATC12 small molecule inhibits the Aurora-A/TPX2 interaction and impairs the proliferation of breast cancer cells

ATC12小分子抑制Aurora-A/TPX2相互作用,从而抑制乳腺癌细胞增殖。

Boi, Dalila; Fianco, Giulia; Polverino, Federica; Fiorentino, Francesco; Mastrangelo, Anna; Rossi, Simone; Rubini, Elisabetta; Rosignoli, Serena; Troilo, Francesca; Antonelli, Maria Rosaria; Tarquini, Dalila; Cervoni, Laura; Rinaldo, Serena; Tramonti, Angela; Scarpone, Eleonora Kristina; Naro, Chiara; Sette, Claudio; Stagni, Venturina; Colotti, Gianni; Rotili, Dante; Paiardini, Alessandro; Guarguaglini, Giulia; Asteriti, Italia Anna

Tumor microenvironment-activated ferritin nanovector enables enhanced tumor delivery of KRAS(G12C) inhibitors and degraders

肿瘤微环境激活的铁蛋白纳米载体可增强KRAS(G12C)抑制剂和降解剂的肿瘤递送。

Abbinantefina, Annalisa Pia; Tito, Claudia; Masciarelli, Silvia; Tisci, Giada; Sortoluzzi, Siria; Ceci, Pierpaolo; Falvo, Elisabetta; Exertier, Cécile; Troilo, Francesca; Petrozza, Vincenzo; Mai, Antonello; Rotili, Dante; Fazi, Francesco; Colotti, Gianni

m(6)A RNA methylation modulates Zika virus infection by regulating serine proteases in Aedes albopictus

m(6)A RNA甲基化通过调节白纹伊蚊中的丝氨酸蛋白酶来调控寨卡病毒感染

Amarante, Anderson de Mendonça; Tirloni, Lucas; Koch, Jonas; Bormann, Felix; Rosignoli, Serena; Paiardini, Alessandro; Rotili, Dante; Brito, Tarcisio; Tavares, Laura de Andrade; Yasumura, Juan Diego de Paula Li; Carneiro, Vitor Coutinho; Kury, Laura Menendez; Pane, Attilio; Lyko, Frank; Fantappié, Marcelo Rosado

Structural snapshots of Pseudomonas aeruginosa LptB(2)FG and LptB(2)FGC reveal insights into lipopolysaccharide recognition and transport.

铜绿假单胞菌 LptB(2)FG 和 LptB(2)FGC 的结构快照揭示了脂多糖识别和运输的见解。

Fiorentino Francesco, Cervoni Matteo, Wang Yi, Urner Leonhard H, Sauer Joshua B, Tran Anh, Corey Robin A, Rotili Dante, Mai Antonello, Stansfeld Phillip J, Imperi Francesco, Yu Edward W, Su Chih-Chia, Robinson Carol V, Bolla Jani R

Activation and inhibition of sirtuins: From bench to bedside

sirtuins 的激活和抑制:从实验室到临床

Fiorentino, Francesco; Fabbrizi, Emanuele; Mai, Antonello; Rotili, Dante

An Amazing 30-Year Journey around the DABO Family: A Medicinal Chemistry Lesson on a Versatile Class of Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors

DABO家族30年奇妙历程:一堂关于多功能非核苷类HIV-1逆转录酶抑制剂的药物化学课

Fabbrizi, Emanuele; Chernyshov, Vladimir V; Fiorentino, Francesco; Sbardella, Gianluca; Ragno, Rino; Nawrozkij, Maxim; Ivanov, Roman; Rotili, Dante; Mai, Antonello

Optimization of Lipoplexes Functionalized with a Sialic Acid Mimetic (F9-PEG) to Target the C1858T PTPN22 Variant for Preclinical Assessment of a Novel Immunotherapy in Endocrine Autoimmunity

利用唾液酸类似物(F9-PEG)功能化的脂质体复合物优化靶向C1858T PTPN22变体,用于内分泌自身免疫新型免疫疗法的临床前评估

Sennato, Simona; Paldino, Giorgia; Bombelli, Cecilia; Mezzani, Irene; Petrini, Stefania; Delfino, Domenico Vittorio; Fiorentino, Francesco; Marianecci, Carlotta; Ciogli, Alessia; Rotili, Dante; Ceccacci, Francesca; Fierabracci, Alessandra

Unraveling the Roles of Epigenetic Regulators During the Embryonic Development of Rhipicephalus microplus

揭示表观遗传调控因子在微小牛蜱胚胎发育中的作用

Amarante, Anderson Mendonça; de Oliveira, Daniel Martins; de Souza, Marcos Paulo Nicolich Camargo; Fonseca-Oliveira, Manoel; Galina, Antonio; Rosignoli, Serena; Arcanjo, Angélica Fernandes; Moraes, Bruno; Paiardini, Alessandro; Rotili, Dante; de Paula Li Yasumura, Juan Diego; Henaut-Jacobs, Sarah; Venancio, Thiago Motta; Uhl, Marcelle; Nunes-da-Fonseca, Rodrigo; Parizi, Luis Fernando; da Silva Vaz Junior, Itabajara; Dos Santos Mermelstein, Claudia; Rios, Thamara; Tirloni, Lucas; Logullo, Carlos; Fantappié, Marcelo Rosado