Optimization of Potent and Selective Cyclohexyl Acid ERAP1 Inhibitors Using Structure- and Property-Based Drug Design
利用基于结构和性质的药物设计优化高效选择性环己酸ERAP1抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.4c00401
Hryczanek, Ross P; Hackett, Andrew S; Rowland, Paul; Chung, Chun-Wa; Convery, Máire A; Holmes, Duncan S; Hutchinson, Jonathan P; Kitchen, Semra; Korczynska, Justyna; Law, Robert P; Lea, Jonathan D; Liddle, John; Lonsdale, Richard; Neu, Margarete; Nickels, Leng; Phillipou, Alex; Rowedder, James E; Schneck, Jessica L; Scott-Stevens, Paul; Sheehan, Hester; Tayler, Chloe L; Temponeras, Ioannis; Tinworth, Christopher P; Walker, Ann L; Wojno-Picon, Justyna; Young, Robert J; Lindsay, David M; Stratikos, Efstratios