Potent and selective bivalent inhibitors of BET bromodomains
强效且选择性的 BET 溴结构域双价抑制剂
期刊:Nature Chemical Biology
影响因子:12.9
doi:10.1038/nchembio.2210
Michael J Waring, Huawei Chen, Alfred A Rabow, Graeme Walker, Romel Bobby, Scott Boiko, Rob H Bradbury, Rowena Callis, Edwin Clark, Ian Dale, Danette L Daniels, Austin Dulak, Liz Flavell, Geoff Holdgate, Thomas A Jowitt, Alexey Kikhney, Mark McAlister, Jacqui Méndez, Derek Ogg, Joe Patel, Philip Pet