TUB-040, a Homogeneous and Hydrophilic NaPi2b-Targeting ADC with Stably Linked Exatecan, Exhibits Long-lasting Antitumor Activity and a Well-Tolerated Safety Profile.
TUB-040 是一种均质亲水性 NaPi2b 靶向 ADC,其稳定连接了依沙替康,具有持久的抗肿瘤活性和良好的耐受性安全性。
期刊:Molecular Cancer Therapeutics
影响因子:5.5
doi:10.1158/1535-7163.MCT-25-0254
Vogl Annette M, Schmitt Saskia, Mai Isabelle, Machui Paul, Herterich Sarah, Leonardi Natascia, Cyprys Philipp, Hauswald Danila, Ochtrop Philipp, Kozlowska Izabela, Kitowski Annabel, Gerlach Marcus, Waldmann Florian, Marcq Olivier, Trail Pamela A, Schumacher Dominik, Fingerle-Rowson Günter R, Hock Björn, Kasper Marc-André, Helma Jonas