日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A guanidine-based coronavirus replication inhibitor which targets the nsp15 endoribonuclease and selects for interferon-susceptible mutant viruses

一种基于胍的冠状病毒复制抑制剂,靶向nsp15核糖核酸内切酶,并筛选出对干扰素敏感的突变病毒。

Van Loy, Benjamin; Pujol, Eugènia; Kamata, Kenichi; Lee, Xiao Yin; Bakirtzoglou, Nikolai; Van Berwaer, Ria; Vandeput, Julie; Mestdagh, Cato; Persoons, Leentje; De Wijngaert, Brent; Goovaerts, Quinten; Noppen, Sam; Jacquemyn, Maarten; Ahmadzadeh, Kourosh; Bernaerts, Eline; Martín-López, Juan; Escriche, Celia; Vanmechelen, Bert; Krasniqi, Besir; Singh, Abhimanyu K; Daelemans, Dirk; Maes, Piet; Matthys, Patrick; Dehaen, Wim; Rozenski, Jef; Das, Kalyan; Voet, Arnout; Vázquez, Santiago; Naesens, Lieve; Stevaert, Annelies

Structure-Activity Relationship Study of 3-Alkynyl-6-aryl-isothiazolo[4,3-b]pyridines as Dual Inhibitors of the Lipid Kinases PIKfyve and PIP4K2C

3-炔基-6-芳基-异噻唑并[4,3-b]吡啶类化合物作为脂质激酶PIKfyve和PIP4K2C双重抑制剂的构效关系研究

Kalebic, Demian; Gao, Ling-Jie; Martinez-Gualda, Belén; Karim, Marwah; Saul, Sirle; Tran, Do Hoang Nhu; Rozenski, Jef; Persoons, Leentje; Schols, Dominique; Dehaen, Wim; Einav, Shirit; De Jonghe, Steven

Tuning i-motif folding and stability with acyclic phosphonate-linked (ZNA) cytidine residues

利用非环状膦酸酯连接的(ZNA)胞嘧啶残基调节i基序的折叠和稳定性

Derden, Marlies; Reynders, Sten; Rihon, Jérôme; Li, Xinlu; Coosemans, Frédérick; Rozenski, Jef; Herdewijn, Piet; Groaz, Elisabetta; Lescrinier, Eveline

Modularity of RBC hitchhiking with polymeric nanoparticles: testing the limits of non-covalent adsorption.

红细胞与聚合物纳米粒子搭便车的模块化:测试非共价吸附的极限

Lenders Vincent, Escudero Remei, Koutsoumpou Xanthippi, Armengol Álvarez Laura, Rozenski Jef, Soenen Stefaan J, Zhao Zongmin, Mitragotri Samir, Baatsen Pieter, Allegaert Karel, Toelen Jaan, Manshian Bella B

Ways to Improve Insights into Clindamycin Pharmacology and Pharmacokinetics Tailored to Practice

提高对克林霉素药理学和药代动力学认识的实践方法

Armengol Álvarez, Laura; Van de Sijpe, Greet; Desmet, Stefanie; Metsemakers, Willem-Jan; Spriet, Isabel; Allegaert, Karel; Rozenski, Jef

Rational design of an XNA ligase through docking of unbound nucleic acids to toroidal proteins

通过将游离核酸对接至环状蛋白,合理设计XNA连接酶

Vanmeert, Michiel; Razzokov, Jamoliddin; Mirza, Muhammad Usman; Weeks, Stephen D; Schepers, Guy; Bogaerts, Annemie; Rozenski, Jef; Froeyen, Mathy; Herdewijn, Piet; Pinheiro, Vitor B; Lescrinier, Eveline

Potential for Biocontrol of Hairy Root Disease by a Paenibacillus Clade

类芽孢杆菌分支对毛状根病生物防治的潜力

Bosmans, Lien; De Bruijn, Irene; Gerards, Saskia; Moerkens, Rob; Van Looveren, Lore; Wittemans, Lieve; Van Calenberge, Bart; Paeleman, Anneleen; Van Kerckhove, Stefan; De Mot, René; Rozenski, Jef; Rediers, Hans; Raaijmakers, Jos M; Lievens, Bart

Synthetic strategy and antiviral evaluation of diamide containing heterocycles targeting dengue and yellow fever virus

合成策略及含二酰胺杂环化合物对登革热病毒和黄热病毒的抗病毒活性评价

Saudi, Milind; Zmurko, Joanna; Kaptein, Suzanne; Rozenski, Jef; Gadakh, Bharat; Chaltin, Patrick; Marchand, Arnaud; Neyts, Johan; Van Aerschot, Arthur

Isothiazolo[4,3-b]pyridines as inhibitors of cyclin G associated kinase : synthesis, structure-activity relationship studies and antiviral activity

异噻唑并[4,3-b]吡啶类化合物作为细胞周期蛋白G相关激酶抑制剂:合成、构效关系研究及抗病毒活性

Li, Jiahong; Kovackova, Sona; Pu, Szuyuan; Rozenski, Jef; De Jonghe, Steven; Einav, Shirit; Herdewijn, Piet

The antimicrobial compound xantholysin defines a new group of Pseudomonas cyclic lipopeptides

抗菌化合物黄素溶素定义了一类新的假单胞菌环状脂肽。

Li, Wen; Rokni-Zadeh, Hassan; De Vleeschouwer, Matthias; Ghequire, Maarten G K; Sinnaeve, Davy; Xie, Guan-Lin; Rozenski, Jef; Madder, Annemieke; Martins, José C; De Mot, René