Peptidylarginine Deiminase (PAD) Inhibitor Optimization through Displacement of a Trapped Water Molecule
通过置换被捕获的水分子来优化肽基精氨酸脱亚胺酶(PAD)抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00372
Schnute, Mark E; Chinigo, Gary M; Futatsugi, Kentaro; Yamaguchi, Masaya; Bagley, Scott W; Banker, Mary Ellen; Chang, Jeanne S; Chen, Ming Z; Choi, Won Young; Corbett, Matthew S; Drozda, Susan E; Ebner, David C; Garcia-Irizarry, Carmen; Hicklin, Robert; Hoy, Susan; Jiao, Wenhua; Kortum, Steven; Lee, Katherine L; Limburg, David C; Lovering, Frank; Moreno, Antonio; Mousseau, James J; Pan, Senliang; Parikh, Mihir D; Pelker, Jeffrey W; Ramsey, Simeon; Reilly, Usa; Rescourio, Gwenaella; Schmitt, Daniel C; Simpson, Brittany; Skrzypek, Grzegorz J; Smaltz, Daniel J; Taylor, Alexandria P; Torella, Rubben; Trujillo, John I; Vajdos, Felix F; Wepy, James A; Wright, Stephen W; Blakemore, David C; Vincent, Fabien; Clerin, Valerie M