Phenotypic Optimization of Urea-Thiophene Carboxamides To Yield Potent, Well Tolerated, and Orally Active Protective Agents against Aminoglycoside-Induced Hearing Loss.
通过表型优化脲噻吩甲酰胺,获得强效、耐受性良好且口服有效的氨基糖苷类药物引起的听力损失保护剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.7b00932
Chowdhury Sarwat, Owens Kelly N, Herr R Jason, Jiang Qin, Chen Xinchao, Johnson Graham, Groppi Vincent E, Raible David W, Rubel Edwin W, Simon Julian A