日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Phase Ia/b Multicenter Study of BPM31510IV Targeting Mitochondrial Metabolism/Warburg Effect as Monotherapy and Combination Chemotherapy in Solid Tumor Patients

BPM31510IV靶向线粒体代谢/瓦博格效应的Ia/b期多中心研究:单药治疗及联合化疗治疗实体瘤患者

Subbiah, Vivek; Yu, Peter P; Sarangarajan, Rangaprasad; Kiebish, Michael A; Rodrigues, Leonardo O; Miller, Gregory M; Akmaev, Viatcheslav R; Luan, Shen; McCook, John P; Tanna, Nikunj; Reilly, Tracey; Chen, Emily; Bussberg, Valerie; Ravipaty, Shobha; Vishnudas, Vivek K; Gesta, Stephane; Lucius, David; Bruce, Can; Hazarika, Suwagmani; Lyng, Arianne; Klotz, Allison; Tolstikov, Vladimir; Stevens, Janice; Chua, Victoria S; Granger, Elder; Tekumalla, Poornima K; Benaim, Ely; Modur, Vijay; Rudoltz, Marc S; Song, Paul Y; Tagawa, Scott T; Hendifer, Andrew; Chawla, Sant P; Shah, Manish A; Hong, David S; Zinner, Ralph; Narain, Niven R; Kundranda, Madappa N

First-in-human study of IM156, a novel potent biguanide oxidative phosphorylation (OXPHOS) inhibitor, in patients with advanced solid tumors

IM156(一种新型强效双胍类氧化磷酸化(OXPHOS)抑制剂)在晚期实体瘤患者中的首次人体研究

Janku, Filip; Beom, Seung-Hoon; Moon, Yong Wha; Kim, Tae Won; Shin, Young G; Yim, Dong-Seok; Kim, Gun Min; Kim, Hyo Song; Kim, Sun Young; Cheong, Jae-Ho; Lee, Young Woo; Geiger, Barb; Yoo, Sanghee; Thurston, Archie; Welsch, Dean; Rudoltz, Marc S; Rha, Sun Young

HGG-40. FOCUSED ULTRASOUND ENHANCES ETOPOSIDE DELIVERY IN A MURINE PONTINE GLIOMA MODEL

HGG-40. 聚焦超声增强依托泊苷在小鼠脑桥胶质瘤模型中的递送

Cannon-Albright, Lisa A; Farnham, James M; Stevens, Jeffrey; Teerlink, Craig C; Palmer, Cheryl A; Rowe, Kerry; Cessna, Melissa H; Blumenthal, Deborah T; Garcia-Moure, Marc; Pérez-Larraya, Jaime Gállego; Patiño, Ana; Gonzalez-Huarriz, Marisol; Jones, Chris; MacKay, Alan; Van der Lugt, Jasper; Hulleman, Esther; de Andrea, Carlos; Astigarraga, Itziar; García-Ariza, Miguel; Lopez-Ibor, Blanca; Villalba, Maria; Lang, Frederick F; Fueyo, Juan; Gomez-Manzano, Candelaria; Dobbs, Jessica; Diez-Valle, Ricardo; Alonso, Marta M; Tejada, Sonia; Seitzman, Benjamin; Anandarajah, Hari; McMichael, Alana; Gu, Hongjie; Barbour, Dennis; Limbrick, David; Shimony, Joshua; Rubin, Joshua; Perkins, Stephanie; Cantor, Evan; Wierzbicki, Kyle; Tarapore, Rohinton S; Thomas, Chase; Cartaxo, Rodrigo; Yadav, Viveka Nand; Ravindran, Ramya; Bruzek, Amy K; Wadden, Jack; Babilla, Clarissa May; Kawakibi, Abed Rhaman; Ji, Sunjong; Ramos, Johanna; Paul, Alyssa; Wolfe, Ian; Leonard, Marcia; Robertson, Partricia; Franson, Andrea; Mody, Rajen; Garton, Hugh; Odia, Yazmin; Kline, Cassie; Vitanza, Nicholas A; Khatua, Soumen; Mueller, Sabine; Allen, Joshua E; Gardner, Sharon; Koschmann, Carl; Leskoske, Kristin; Garcia-Mansfield, Krystine; Krishnan, Aparna; Sharma, Ritin; Rusert, Jessica; Mesirov, Jill; Wechsler-Reya, Robert; Pirrotte, Patrick; Olga, Zheludkova; Liudmila, Olkhova; Ludmilla, Zubarovskaya; Julia, Dinikina; Anna, Smirnova; Yuri, Kushel’; Armenak, Melikyan; Shavkat, Kadyrov; Marina, Ryzhova; Liudmila, Shishkina; Alexey, Kislyakov; Evgeniy, Shultz; Svetlana, Gorbatykh; Olga, Polushkina; Eugenia, Inyushkina; Natalia, Yudina; Asmik, Gevorgian; Liudmila, Privalova; Liudmila, Minkina; Artem, Zaichikov; Ivan, Fisyun; Daniil, Sakun; Vyacheslav, Mitrofanov; Sergey, Kovalenko; Ekaterina, Grishina; Nadezhda, Pishchaeva; Nikolay, Vorob’ev; Nadezhda, Plakhotina; Natalia, Popova; Dmitriy, Pogorelov; Alexander, Shapochnik; Andrey, Korchunov; Zhang, Wenqiu; Mohammad, Afroz; Sirianni, Rachael; Elmquist, William; Abuarqoub, Alqassem; McAnulty, Tatiana; Amiel, Eyal; Stafford, James; Wei, Xin; Phoenix, Timothy; Chi, Susan; Hsieh, Antony; Foley, Megan; Shi, Hongliang; Swamy, Preethi; Rodstrom, Jill; Rudoltz, Marc; Borsuk, Robyn; Zhou, Lanlan; Chang, Wen-i; Zhang, Yiqun; Prabhu, Varun; Allen, Joshua; Tapinos, Nikos; Lulla, Rishi; El-Deiry, Wafik; Moreira, Daniel; Spiller, Susan; Bouldin, Thomas; Davidson, Alan; Saba-Silva, Nasjla; Sullivan, Daniel; Tanaka, Ryuma; Wagner, Aaron; Wood, Matthew; Gajjar, Amar; Chiang, Jason; Maaz, Ata; Yousif, Tayseer; Abdulmajeed, Mohammed; Ederies, Moegamad; Neri, Pedro; Kamboh, Abdul; Silverman, Mackenzie; Piatt, Joseph; Walter, Andrew; Nikam, Rahul; Kaur, Gurcharanjeet; Cosentino, Chiara Cianciolo; Laternser, Sandra; Przystal, Justyna M; Yadavilli, Sridevi; Zhang, Jie; Müller, Timothy; Kritzer, Bettina; Müller, Sabine; Nazarian, Javad; P.Y. Liu, Anthony; Ku, Dennis T L; Fu, Eric; Luk, Chung-Wing; Yau, Jeffrey P W; Ling, Siu-Cheung; Chan, Godfrey C F; Shing, Matthew M K; Park, Hannah; Kobritz, Naomi; Mehdikhani, Shaunt; Breunig, Joshua; Cocito, Carolina; Branchtein, Mylene; Gongora, Tatyana; Dahmane, Nadia; Greenfield, Jeffrey; McSwain, Leon; Kenney, Anna; Chen, Victor; Huang, Tiffany; McNutt, Sarah; Shah, Nidhi; Rizk, Elias; Dennis, T L Ku; Liu, Anthony P Y; Fu, Eric; Luk, Chung-Wing; Yau, Jeffrey P W; Ling, Siu-Cheung; Shing, Matthew M K; Chan, Godfrey C F; Thompson, Dean; Castle, Jemma; Hicks, Debbie; Clifford, Steve; Schwalbe, Ed; Englander, Zachary; Wei, Hong-Jian; Pouliopoulos, Antonios; Yoh, Nina; McQuillan, Nicholas; Tazhibi, Masih; Wang, Tony; Bruce, Jeffrey; Canoll, Peter; Feldstein, Neil; Zacharoulis, Stergios; Konofagou, Elisa; Wu, Cheng-Chia

Repression of LKB1 by miR-17∼92 Sensitizes MYC-Dependent Lymphoma to Biguanide Treatment

miR-17∼92 对 LKB1 的抑制作用使 MYC 依赖性淋巴瘤对双胍类药物治疗更加敏感

Said Izreig ,Alexandra Gariepy ,Irem Kaymak ,Hannah R Bridges ,Ariel O Donayo ,Gaëlle Bridon ,Lisa M DeCamp ,Susan M Kitchen-Goosen ,Daina Avizonis ,Ryan D Sheldon ,Rob C Laister ,Mark D Minden ,Nathalie A Johnson ,Thomas F Duchaine ,Marc S Rudoltz ,Sanghee Yoo ,Michael N Pollak ,Kelsey S Williams ,Russell G Jones

A Direct Comparison of in Vitro and in Vivo Nucleic Acid Delivery Mediated by Hundreds of Nanoparticles Reveals a Weak Correlation

数百个纳米粒子介导的体内和体外核酸输送的直接比较揭示了弱相关性

Kalina Paunovska, Cory D Sago, Christopher M Monaco, William H Hudson, Marielena Gamboa Castro, Tobi G Rudoltz, Sujay Kalathoor, Daryll A Vanover, Philip J Santangelo, Rafi Ahmed, Anton V Bryksin, James E Dahlman

High-throughput in vivo screen of functional mRNA delivery identifies nanoparticles for endothelial cell gene editing

高通量体内筛选功能性mRNA递送纳米颗粒,用于内皮细胞基因编辑

Sago, Cory D; Lokugamage, Melissa P; Paunovska, Kalina; Vanover, Daryll A; Monaco, Christopher M; Shah, Nirav N; Gamboa Castro, Marielena; Anderson, Shannon E; Rudoltz, Tobi G; Lando, Gwyneth N; Munnilal Tiwari, Pooja; Kirschman, Jonathan L; Willett, Nick; Jang, Young C; Santangelo, Philip J; Bryksin, Anton V; Dahlman, James E

Probing the potential of mucus permeability to signify preterm birth risk

探究黏液通透性在预测早产风险方面的潜在作用

Smith-Dupont, K B; Wagner, C E; Witten, J; Conroy, K; Rudoltz, H; Pagidas, K; Snegovskikh, V; House, M; Ribbeck, K

Phase III, randomized, open-label study of daily imatinib mesylate 400 mg versus 800 mg in patients with newly diagnosed, previously untreated chronic myeloid leukemia in chronic phase using molecular end points: tyrosine kinase inhibitor optimization and selectivity study

一项III期随机、开放标签研究,比较每日服用400 mg甲磺酸伊马替尼与800 mg甲磺酸伊马替尼治疗新诊断、既往未接受治疗的慢性期慢性粒细胞白血病患者的疗效,采用分子终点指标:酪氨酸激酶抑制剂优化和选择性研究。

Cortes, Jorge E; Baccarani, Michele; Guilhot, François; Druker, Brian J; Branford, Susan; Kim, Dong-Wook; Pane, Fabrizio; Pasquini, Ricardo; Goldberg, Stuart L; Kalaycio, Matt; Moiraghi, Beatriz; Rowe, Jacob M; Tothova, Elena; De Souza, Carmino; Rudoltz, Marc; Yu, Richard; Krahnke, Tillmann; Kantarjian, Hagop M; Radich, Jerald P; Hughes, Timothy P

Efficacy of imatinib dose escalation in patients with chronic myeloid leukemia in chronic phase

伊马替尼剂量递增治疗慢性期慢性粒细胞白血病患者的疗效

Kantarjian, Hagop M; Larson, Richard A; Guilhot, Francois; O'Brien, Stephen G; Mone, Manisha; Rudoltz, Marc; Krahnke, Tillmann; Cortes, Jorge; Druker, Brian J