日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Multiple intramolecular triggers converge to preferential G protein coupling in the CB(2)R

多种分子内触发因素汇聚于CB(2)受体中G蛋白的优先偶联。

Morales-Pastor, Adrian; Miljuš, Tamara; Dieguez-Eceolaza, Miguel; Stępniewski, Tomasz Maciej; Ledesma-Martin, Vicente; Heydenreich, Franziska M; Flock, Tilman; Plouffe, Bianca; Le Gouill, Christian; Duchaine, Jean; Sykes, David A; Nicholson, Colin; Koers, Eline J; Guba, Wolfgang; Rufer, Arne C; Grether, Uwe; Bouvier, Michel; Veprintsev, Dmitry B; Selent, Jana

CellEKT: A Robust Chemical Proteomics Workflow to Profile Cellular Target Engagement of Kinase Inhibitors.

CellEKT:一种稳健的化学蛋白质组学工作流程,用于分析激酶抑制剂的细胞靶标结合情况

Rüegger Joel, Gagestein Berend, Janssen Antonius P A, Valeanu Alexandra, Mori Alger Lazo, van der Peet Marielle, Boutkan Michael S, Florea Bogdan I, Henneman Alex A, Hochstrasser Remo, Wang Haiyan, Westwood Paul, Topp Andreas, Gomez Barila Patricia M, Medema Jan Paul, Jimenez Connie R, Woersdoerfer Bigna, Kirchner Stephan, Zhang Jitao David, Grether Uwe, Rufer Arne C, van der Stelt Mario

A universal cannabinoid CB1 and CB2 receptor TR-FRET kinetic ligand-binding assay.

一种通用的大麻素 CB1 和 CB2 受体 TR-FRET 动力学配体结合测定法

Borrega-Roman Leire, Hoare Bradley L, Kosar Miroslav, Sarott Roman C, Patej Kacper J, Bouma Jara, Scott-Dennis Morgan, Koers Eline J, Gazzi Thais, Mach Leonard, Barrondo Sergio, Sallés Joan, Guba Wolfgang, Kusznir Eric, Nazaré Marc, Rufer Arne C, Grether Uwe, Heitman Laura H, Carreira Erick M, Sykes David A, Veprintsev Dmitry B

Biased Signaling and Its Role in the Genesis of Short- and Long-Acting β(2)-Adrenoceptor Agonists.

偏向性信号传导及其在短效和长效β2-肾上腺素受体激动剂产生中的作用

Phan Ngan T N, Borrega-Roman Leire, Hoare Bradley L, Harwood Clare R, Geary Natalie, Guba Wolfgang, Han Yongqi, Zenko Vladimirs, Koers Eline J, Rufer Arne C, Grether Uwe, Veprintsev Dmitry B, Sykes David A

Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe

利用高效、细胞渗透性荧光探针检测天然细胞和斑马鱼中的大麻素受体2型

Gazzi, Thais; Brennecke, Benjamin; Atz, Kenneth; Korn, Claudia; Sykes, David; Forn-Cuni, Gabriel; Pfaff, Patrick; Sarott, Roman C; Westphal, Matthias V; Mostinski, Yelena; Mach, Leonard; Wasinska-Kalwa, Malgorzata; Weise, Marie; Hoare, Bradley L; Miljuš, Tamara; Mexi, Maira; Roth, Nicolas; Koers, Eline J; Guba, Wolfgang; Alker, André; Rufer, Arne C; Kusznir, Eric A; Huber, Sylwia; Raposo, Catarina; Zirwes, Elisabeth A; Osterwald, Anja; Pavlovic, Anto; Moes, Svenja; Beck, Jennifer; Nettekoven, Matthias; Benito-Cuesta, Irene; Grande, Teresa; Drawnel, Faye; Widmer, Gabriella; Holzer, Daniela; van der Wel, Tom; Mandhair, Harpreet; Honer, Michael; Fingerle, Jürgen; Scheffel, Jörg; Broichhagen, Johannes; Gawrisch, Klaus; Romero, Julián; Hillard, Cecilia J; Varga, Zoltan V; van der Stelt, Mario; Pacher, Pal; Gertsch, Jürg; Ullmer, Christoph; McCormick, Peter J; Oddi, Sergio; Spaink, Herman P; Maccarrone, Mauro; Veprintsev, Dmitry B; Carreira, Erick M; Grether, Uwe; Nazaré, Marc

Reply to Alarcon and Borroto: Small molecule AX-024 reduces T cell proliferation independently of CD3ε-Nck1 interaction at SH3.1

回复 Alarcon 和 Borroto:小分子 AX-024 可降低 T 细胞增殖,且该作用独立于 SH3.1 位点的 CD3ε-Nck1 相互作用。

Richter, Kirsten; Rufer, Arne C; Muller, Magali; Burger, Dominique; Casagrande, Fabio; Grossenbacher, Tabea; Huber, Sylwia; Hug, Melanie N; Koldewey, Philipp; D'Osualdo, Andrea; Schlatter, Daniel; Stoll, Theodor; Rudolph, Markus G

A multilaboratory comparison of calibration accuracy and the performance of external references in analytical ultracentrifugation

分析超速离心中校准精度和外部参考性能的多实验室比较

Zhao, Huaying; Ghirlando, Rodolfo; Alfonso, Carlos; Arisaka, Fumio; Attali, Ilan; Bain, David L; Bakhtina, Marina M; Becker, Donald F; Bedwell, Gregory J; Bekdemir, Ahmet; Besong, Tabot M D; Birck, Catherine; Brautigam, Chad A; Brennerman, William; Byron, Olwyn; Bzowska, Agnieszka; Chaires, Jonathan B; Chaton, Catherine T; Cölfen, Helmut; Connaghan, Keith D; Crowley, Kimberly A; Curth, Ute; Daviter, Tina; Dean, William L; Díez, Ana I; Ebel, Christine; Eckert, Debra M; Eisele, Leslie E; Eisenstein, Edward; England, Patrick; Escalante, Carlos; Fagan, Jeffrey A; Fairman, Robert; Finn, Ron M; Fischle, Wolfgang; de la Torre, José García; Gor, Jayesh; Gustafsson, Henning; Hall, Damien; Harding, Stephen E; Cifre, José G Hernández; Herr, Andrew B; Howell, Elizabeth E; Isaac, Richard S; Jao, Shu-Chuan; Jose, Davis; Kim, Soon-Jong; Kokona, Bashkim; Kornblatt, Jack A; Kosek, Dalibor; Krayukhina, Elena; Krzizike, Daniel; Kusznir, Eric A; Kwon, Hyewon; Larson, Adam; Laue, Thomas M; Le Roy, Aline; Leech, Andrew P; Lilie, Hauke; Luger, Karolin; Luque-Ortega, Juan R; Ma, Jia; May, Carrie A; Maynard, Ernest L; Modrak-Wojcik, Anna; Mok, Yee-Foong; Mücke, Norbert; Nagel-Steger, Luitgard; Narlikar, Geeta J; Noda, Masanori; Nourse, Amanda; Obsil, Tomas; Park, Chad K; Park, Jin-Ku; Pawelek, Peter D; Perdue, Erby E; Perkins, Stephen J; Perugini, Matthew A; Peterson, Craig L; Peverelli, Martin G; Piszczek, Grzegorz; Prag, Gali; Prevelige, Peter E; Raynal, Bertrand D E; Rezabkova, Lenka; Richter, Klaus; Ringel, Alison E; Rosenberg, Rose; Rowe, Arthur J; Rufer, Arne C; Scott, David J; Seravalli, Javier G; Solovyova, Alexandra S; Song, Renjie; Staunton, David; Stoddard, Caitlin; Stott, Katherine; Strauss, Holger M; Streicher, Werner W; Sumida, John P; Swygert, Sarah G; Szczepanowski, Roman H; Tessmer, Ingrid; Toth, Ronald T 4th; Tripathy, Ashutosh; Uchiyama, Susumu; Uebel, Stephan F W; Unzai, Satoru; Gruber, Anna Vitlin; von Hippel, Peter H; Wandrey, Christine; Wang, Szu-Huan; Weitzel, Steven E; Wielgus-Kutrowska, Beata; Wolberger, Cynthia; Wolff, Martin; Wright, Edward; Wu, Yu-Sung; Wubben, Jacinta M; Schuck, Peter

Isothermal titration calorimetry with micelles: Thermodynamics of inhibitor binding to carnitine palmitoyltransferase 2 membrane protein

利用胶束等温滴定量热法:抑制剂与肉碱棕榈酰转移酶2膜蛋白结合的热力学研究

Perspicace, Samantha; Rufer, Arne C; Thoma, Ralf; Mueller, Francis; Hennig, Michael; Ceccarelli, Simona; Schulz-Gasch, Tanja; Seelig, Joachim

Structural insight into function and regulation of carnitine palmitoyltransferase

肉碱棕榈酰转移酶的功能和调控的结构解析

Rufer, Arne C; Thoma, Ralf; Hennig, Michael