Discovery of LC-MI-3: A Potent and Orally Bioavailable Degrader of Interleukin-1 Receptor-Associated Kinase 4 for the Treatment of Inflammatory Diseases
发现 LC-MI-3:一种有效且口服生物可利用的白细胞介素-1 受体相关激酶 4 降解剂,可用于治疗炎症疾病
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c00181
Lingfeng Chen, Ruixiang Luo, Lin Ma, Ying Xu, Jiaqi Cao, Zheng Jiang, Shiyan Chen, Xiaohao Huang, Mingwan Zhang, Lei Zheng, Yawen Zhang, Lina Yin, Jie Yu, Xiaochun Zheng, Lulu Zheng, Ping Huang, Guang Liang