日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Blockade of the MEK/ERK signalling cascade by AS703026, a novel selective MEK1/2 inhibitor, induces pleiotropic anti-myeloma activity in vitro and in vivo

AS703026(一种新型选择性 MEK1/2 抑制剂)可阻断 MEK/ERK 信号级联,从而在体外和体内诱导多效性抗骨髓瘤活性

Kihyun Kim, Sun-Young Kong, Mariateresa Fulciniti, Xianfeng Li, Weihua Song, Sabikun Nahar, Peter Burger, Mathew J Rumizen, Klaus Podar, Dharminder Chauhan, Teru Hideshima, Nikhil C Munshi, Paul Richardson, Ann Clark, Janet Ogden, Andreas Goutopoulos, Luca Rastelli, Kenneth C Anderson, Yu-Tzu Tai

CS1 promotes multiple myeloma cell adhesion, clonogenic growth, and tumorigenicity via c-maf-mediated interactions with bone marrow stromal cells

CS1通过c-maf介导的与骨髓基质细胞的相互作用,促进多发性骨髓瘤细胞的黏附、克隆形成和致瘤性。

Tai, Yu-Tzu; Soydan, Ender; Song, Weihua; Fulciniti, Mariateresa; Kim, Kihyun; Hong, Fangxin; Li, Xian-Feng; Burger, Peter; Rumizen, Matthew J; Nahar, Sabikun; Podar, Klaus; Hideshima, Teru; Munshi, Nikhil C; Tonon, Giovanni; Carrasco, Ruben D; Afar, Daniel E H; Anderson, Kenneth C