Blockade of the MEK/ERK signalling cascade by AS703026, a novel selective MEK1/2 inhibitor, induces pleiotropic anti-myeloma activity in vitro and in vivo
AS703026(一种新型选择性 MEK1/2 抑制剂)可阻断 MEK/ERK 信号级联,从而在体外和体内诱导多效性抗骨髓瘤活性
期刊:British Journal of Haematology
影响因子:5.1
doi:10.1111/j.1365-2141.2010.08127.x
Kihyun Kim, Sun-Young Kong, Mariateresa Fulciniti, Xianfeng Li, Weihua Song, Sabikun Nahar, Peter Burger, Mathew J Rumizen, Klaus Podar, Dharminder Chauhan, Teru Hideshima, Nikhil C Munshi, Paul Richardson, Ann Clark, Janet Ogden, Andreas Goutopoulos, Luca Rastelli, Kenneth C Anderson, Yu-Tzu Tai