日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The immunological and pharmacokinetic evaluation of Lipid-PLGA hybrid nanoparticle-based oxycodone vaccines

基于脂质-PLGA杂化纳米颗粒的羟考酮疫苗的免疫学和药代动力学评价

Walter, Debra L; Bian, Yuanzhi; Hu, He; Hamid, Fatima A; Rostamizadeh, Kobra; Vigliaturo, Jennifer R; DeHority, Riley; Ehrich, Marion; Runyon, Scott; Pravetoni, Marco; Zhang, Chenming

Bivalent Hapten Display Strategies for Conjugate Vaccines Targeting Opioid Mixtures Containing Fentanyl

针对含芬太尼阿片类药物混合物的结合疫苗的二价半抗原展示策略

Baehr, Carly; Jahan, Rajwana; Gebo, Ann; Vigliaturo, Jennifer; Song, Daihyun; Rahman, Md Toufiqur; Tronconi, Davide; Khaimraj, Aaron; Seaman, Robert; Marecki, Courtney; Kim, Caroline M; Persano, Stefano; Runyon, Scott P; Pravetoni, Marco

Indazole partial agonists targeting peripheral cannabinoid receptors

靶向外周大麻素受体的吲唑类部分激动剂

Amato, George; Laudermilk, Lucas; Vasukuttan, Vineetha; Gay, Elaine A; Decker, Ann M; Snyder, Rodney; Yue, Yun Lan; Runyon, Scott; Maitra, Rangan

A humanized monoclonal antibody attenuates carfentanil self-administration in nonhuman primates

人源化单克隆抗体可减弱非人灵长类动物对卡芬太尼的自我给药行为

Galbo-Thomma, Lindsey K; Baehr, Carly; Gay, Elaine A; Runyon, Scott; Pravetoni, Marco; France, Charles P

The Influence of the Estrous Cycle on Neuropeptide S Receptor-Mediated Behaviors

动情周期对神经肽S受体介导行为的影响

Costa, Paula Carvalho; Salinas, Brisa; Wojciechowski, Alaina; Wood, Susan K; Runyon, Scott; Clark, Stewart D

Studies on diketopiperazine and dipeptide analogs as opioid receptor ligands

二酮哌嗪和二肽类似物作为阿片受体配体的研究

Shahbazi Nia, Siavash; Hossain, Mohammad Anwar; Ji, Guangchen; Jonnalagadda, Sravan K; Obeng, Samuel; Rahman, Md Ashrafur; Sifat, Ali Ehsan; Nozohouri, Saeideh; Blackwell, Collin; Patel, Dhavalkumar; Thompson, Jon; Runyon, Scott; Hiranita, Takato; McCurdy, Christopher R; McMahon, Lance; Abbruscato, Thomas J; Trippier, Paul C; Neugebauer, Volker; German, Nadezhda A

Structures of drug-specific monoclonal antibodies bound to opioids and nicotine reveal a common mode of binding.

与阿片类药物和尼古丁结合的药物特异性单克隆抗体的结构揭示了一种共同的结合模式

Rodarte Justas V, Baehr Carly, Hicks Dustin, Liban Tyler L, Weidle Connor, Rupert Peter B, Jahan Rajwana, Wall Abigail, McGuire Andrew T, Strong Roland K, Runyon Scott, Pravetoni Marco, Pancera Marie

Discovery of 1,3-disubstituted pyrazole peripheral cannabinoid receptor partial agonists

1,3-二取代吡唑外周大麻素受体部分激动剂的发现

Amato, George; Runyon, Scott; Vasukuttan, Vineetha; Decker, Ann M; Gay, Elaine A; Laudermilk, Lucas; Maitra, Rangan

Structure-Activity Relationship Development Efforts towards Peripherally Selective Analogs of the Cannabinoid Receptor Partial Agonist BAY 59-3074

针对大麻素受体部分激动剂 BAY 59-3074 的外周选择性类似物的结构-活性关系研究

Amato, George; Vasukuttan, Vineetha; Harris, Danni; Laudermilk, Lucas; Lucitti, Jennifer; Runyon, Scott; Maitra, Rangan

Preclinical Efficacy and Selectivity of Vaccines Targeting Fentanyl, Alfentanil, Sufentanil, and Acetylfentanyl in Rats

芬太尼、阿芬太尼、舒芬太尼和乙酰芬太尼靶向疫苗在大鼠中的临床前疗效和选择性

Baehr, Carly; Robinson, Christine; Kassick, Andrew; Jahan, Rajwana; Gradinati, Valeria; Averick, Saadyah E; Runyon, Scott P; Pravetoni, Marco