日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A robust fluorogenic substrate for chikungunya virus protease (nsP2) activity

一种用于检测基孔肯雅病毒蛋白酶(nsP2)活性的强效荧光底物

Makhaik, Sparsh; Rut, Wioletta; Choudhary, Shruti; Upadhyay, Tulsi; Hao, Chenzhou; Westberg, Michael; Bobst, Cedric; Yoo, Euna; Fejzo, Jasna; Lin, Michael Z; Bogyo, Matthew; Thompson, Paul; Drag, Marcin; Hardy, Jeanne A

A Robust Fluorogenic Substrate for Chikungunya Virus Protease (nsP2) Activity

一种用于检测基孔肯雅病毒蛋白酶 (nsP2) 活性的强效荧光底物

Makhaik, Sparsh; Rut, Wioletta; Choudhary, Shruti; Upadhyay, Tulsi; Hao, Chenzhou; Westberg, Michael; Bobst, Cedric; Yoo, Euna; Fejzo, Jasna; Lin, Michael Z; Bogyo, Matthew; Thompson, Paul; Drag, Marcin; Hardy, Jeanne A

Profiling of coronaviral M(pro) and enteroviral 3C(pro) specificity provides a framework for the development of broad-spectrum antiviral compounds

对冠状病毒M蛋白和肠道病毒3C蛋白特异性的分析为开发广谱抗病毒化合物提供了框架。

Rut, Wioletta; Groborz, Katarzyna; Sun, Xinyuanyuan; Hilgenfeld, Rolf; Drag, Marcin

Use of protease substrate specificity screening in the rational design of selective protease inhibitors with unnatural amino acids: Application to HGFA, matriptase, and hepsin.

利用蛋白酶底物特异性筛选合理设计含非天然氨基酸的选择性蛋白酶抑制剂:应用于 HGFA、matriptase 和 hepsin

Mahoney Matthew W, Helander Jonathan, Kooner Anoopjit S, Norman Mariah, Damalanka Vishnu C, De Bona Paolo, Kasperkiewicz Paulina, Rut Wioletta, Poreba Marcin, Kashipathy Maithri M, Battaile Kevin P, Lovell Scott, O'Donoghue Anthony J, Craik Charles S, Drag Marcin, Janetka James W

SARS-CoV-2 M(pro) Protease Variants of Concern Display Altered Viral Substrate and Cell Host Target Galectin-8 Processing but Retain Sensitivity toward Antivirals

值得关注的SARS-CoV-2 M(pro)蛋白酶变体表现出病毒底物和细胞宿主靶标半乳糖凝集素-8加工的改变,但仍对抗菌药物敏感

Chen, Sizhu Amelia; Arutyunova, Elena; Lu, Jimmy; Khan, Muhammad Bashir; Rut, Wioletta; Zmudzinski, Mikolaj; Shahbaz, Shima; Iyyathurai, Jegan; Moussa, Eman W; Turner, Zoe; Bai, Bing; Lamer, Tess; Nieman, James A; Vederas, John C; Julien, Olivier; Drag, Marcin; Elahi, Shokrollah; Young, Howard S; Lemieux, M Joanne

Activity profiling and crystal structures of inhibitor-bound SARS-CoV-2 papain-like protease: A framework for anti-COVID-19 drug design

抑制剂结合的SARS-CoV-2木瓜蛋白酶样蛋白酶的活性分析和晶体结构:抗COVID-19药物设计的框架

Rut, Wioletta; Lv, Zongyang; Zmudzinski, Mikolaj; Patchett, Stephanie; Nayak, Digant; Snipas, Scott J; El Oualid, Farid; Huang, Tony T; Bekes, Miklos; Drag, Marcin; Olsen, Shaun K

Counter Selection Substrate Library Strategy for Developing Specific Protease Substrates and Probes.

反向选择底物库策略用于开发特异性蛋白酶底物和探针

Poreba Marcin, Solberg Rigmor, Rut Wioletta, Lunde Ngoc Nguyen, Kasperkiewicz Paulina, Snipas Scott J, Mihelic Marko, Turk Dusan, Turk Boris, Salvesen Guy S, Drag Marcin

Small Molecule Active Site Directed Tools for Studying Human Caspases

用于研究人类半胱天冬酶的小分子活性位点靶向工具

Poreba, Marcin; Szalek, Aleksandra; Kasperkiewicz, Paulina; Rut, Wioletta; Salvesen, Guy S; Drag, Marcin

SARS hCoV papain-like protease is a unique Lys48 linkage-specific di-distributive deubiquitinating enzyme

SARS hCoV 木瓜蛋白酶样蛋白酶是一种独特的 Lys48 连接特异性双分布去泛素化酶

Békés, Miklós; Rut, Wioletta; Kasperkiewicz, Paulina; Mulder, Monique P C; Ovaa, Huib; Drag, Marcin; Lima, Christopher D; Huang, Tony T