Targeting the ERα DBD-LBD Interface with Mitoxantrone Disrupts Receptor Function through Proteasomal Degradation.
利用米托蒽醌靶向 ERα DBD-LBD 界面,通过蛋白酶体降解破坏受体功能。
期刊:Molecular Cancer Therapeutics
影响因子:5.5
doi:10.1158/1535-7163.MCT-25-0405
Wang Han, Luo Yuxuan, Artham Sandeep, Wang Qianqian, Peng Yi, Yun Zixi, Li Xinyue, Wu Chen, Liu Zhenghao, Weber-Bonk Kristen L, Pai Chun-Peng, Cao Yuan, Yue Jiangan, Park Sunghee, Keri Ruth A, Geng Lisheng, McDonnell Donald P, Kao Hung-Ying, Yang Sichun