Zampanolide, a potent new microtubule-stabilizing agent, covalently reacts with the taxane luminal site in tubulin α,β-heterodimers and microtubules
Zampanolide 是一种新型强效微管稳定剂,可与微管蛋白 α、β-异二聚体和微管中的紫杉烷腔内位点发生共价反应
期刊:Chemistry & Biology
影响因子:
doi:10.1016/j.chembiol.2012.05.008
Jessica J Field, Benet Pera, Enrique Calvo, Angeles Canales, Didier Zurwerra, Chiara Trigili, Javier Rodríguez-Salarichs, Ruth Matesanz, Arun Kanakkanthara, St John Wakefield, A Jonathan Singh, Jesús Jiménez-Barbero, Peter Northcote, John H Miller, Juan Antonio López, Ernest Hamel, Isabel Barasoain,