日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Orthosteric STING inhibition elucidates molecular correction of SAVI STING.

正构 STING 抑制阐明了 SAVI STING 的分子矫正

Xie Tao, Ruzanov Max, Critton David, Merselis Leidy, Naglich Joseph, Sack John S, Zhang Ping, Xie Chunshan, Tredup Jeffrey, Stine Laurel B, Messier Cameron, Hope David L, Caceres-Cortes Janet, Mueller Luciano, Dyckman Alaric J, Newitt John A, Choudhury Asmita, Wilson Stephen C

Azatricyclic Inverse Agonists of RORγt That Demonstrate Efficacy in Models of Rheumatoid Arthritis and Psoriasis

在类风湿性关节炎和银屑病模型中显示出疗效的RORγt氮杂三环反向激动剂

Liu, Qingjie; Xiao, Hai-Yun; Batt, Douglas G; Xiao, Zili; Zhu, Yeheng; Yang, Michael G; Li, Ning; Yip, Shiuhang; Li, Peng; Sun, Dawn; Wu, Dauh-Rurng; Ruzanov, Max; Sack, John S; Weigelt, Carolyn A; Wang, Jinhong; Li, Sha; Shuster, David J; Xie, Jenny H; Song, Yunling; Sherry, Tara; Obermeier, Mary T; Fura, Aberra; Stefanski, Kevin; Cornelius, Georgia; Chacko, Silvi; Khandelwal, Purnima; Dudhgaonkar, Shailesh; Rudra, Anjuman; Nagar, Jignesh; Murali, Venkata; Govindarajan, Arun; Denton, Rex; Zhao, Qihong; Meanwell, Nicholas A; Borzilleri, Robert; Dhar, T G Murali

Using yeast surface display to engineer a soluble and crystallizable construct of hematopoietic progenitor kinase 1 (HPK1)

利用酵母表面展示技术构建可溶且可结晶的造血祖细胞激酶 1 (HPK1) 结构

Lau, Wai L; Pearce, Bradley; Malakian, Heather; Rodrigo, Iyoncy; Xie, Dianlin; Gao, Mian; Marsilio, Frank; Chang, Chiehying; Ruzanov, Max; Muckelbauer, Jodi K; Newitt, John A; Lipovšek, Daša; Sheriff, Steven

Discovery of BMS-986251: A Clinically Viable, Potent, and Selective RORγt Inverse Agonist

BMS-986251 的发现:一种临床上可行、高效且选择性的 RORγt 反向激动剂

Cherney, Robert J; Cornelius, Lyndon A M; Srivastava, Anurag; Weigelt, Carolyn A; Marcoux, David; Duan, James J-W; Shi, Qing; Batt, Douglas G; Liu, Qingjie; Yip, Shiuhang; Wu, Dauh-Rurng; Ruzanov, Max; Sack, John; Khan, Javed; Wang, Jinhong; Yarde, Melissa; Cvijic, Mary Ellen; Mathur, Arvind; Li, Sha; Shuster, David; Khandelwal, Purnima; Borowski, Virna; Xie, Jenny; Obermeier, Mary; Fura, Aberra; Stefanski, Kevin; Cornelius, Georgia; Tino, Joseph A; Macor, John E; Salter-Cid, Luisa; Denton, Rex; Zhao, Qihong; Carter, Percy H; Dhar, T G Murali

Discovery of BMS-986260, a Potent, Selective, and Orally Bioavailable TGFβR1 Inhibitor as an Immuno-oncology Agent

发现强效、选择性强且口服生物利用度高的TGFβR1抑制剂BMS-986260,可作为免疫肿瘤药物

Velaparthi, Upender; Darne, Chetan Padmakar; Warrier, Jayakumar; Liu, Peiying; Rahaman, Hasibur; Augustine-Rauch, Karen; Parrish, Karen; Yang, Zheng; Swanson, Jesse; Brown, Jennifer; Dhar, Gopal; Anandam, Aravind; Holenarsipur, Vinay K; Palanisamy, Kamalavenkatesh; Wautlet, Barri S; Fereshteh, Mark P; Lippy, Jonathan; Tebben, Andrew J; Sheriff, Steven; Ruzanov, Max; Yan, Chunhong; Gupta, Anuradha; Gupta, Arun Kumar; Vetrichelvan, Muthalagu; Mathur, Arvind; Gelman, Marina; Singh, Rajinder; Kinsella, Todd; Murtaza, Anwar; Fargnoli, Joseph; Vite, Gregory; Borzilleri, Robert M

Discovery of 4-Azaindole Inhibitors of TGFβRI as Immuno-oncology Agents

发现 4-氮杂吲哚类 TGFβRI 抑制剂作为免疫肿瘤药物

Zhang, Yong; Zhao, Yufen; Tebben, Andrew J; Sheriff, Steven; Ruzanov, Max; Fereshteh, Mark P; Fan, Yi; Lippy, Jonathan; Swanson, Jesse; Ho, Ching-Ping; Wautlet, Barri S; Rose, Anne; Parrish, Karen; Yang, Zheng; Donnell, Andrew F; Zhang, Liping; Fink, Brian E; Vite, Gregory D; Augustine-Rauch, Karen; Fargnoli, Joseph; Borzilleri, Robert M