Azatricyclic Inverse Agonists of RORγt That Demonstrate Efficacy in Models of Rheumatoid Arthritis and Psoriasis
在类风湿性关节炎和银屑病模型中显示出疗效的RORγt氮杂三环反向激动剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.1c00112
Liu, Qingjie; Xiao, Hai-Yun; Batt, Douglas G; Xiao, Zili; Zhu, Yeheng; Yang, Michael G; Li, Ning; Yip, Shiuhang; Li, Peng; Sun, Dawn; Wu, Dauh-Rurng; Ruzanov, Max; Sack, John S; Weigelt, Carolyn A; Wang, Jinhong; Li, Sha; Shuster, David J; Xie, Jenny H; Song, Yunling; Sherry, Tara; Obermeier, Mary T; Fura, Aberra; Stefanski, Kevin; Cornelius, Georgia; Chacko, Silvi; Khandelwal, Purnima; Dudhgaonkar, Shailesh; Rudra, Anjuman; Nagar, Jignesh; Murali, Venkata; Govindarajan, Arun; Denton, Rex; Zhao, Qihong; Meanwell, Nicholas A; Borzilleri, Robert; Dhar, T G Murali