日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Design of a Chemical Probe Set for the 5-HT5A Serotonin Receptor

基于结构设计 5-HT5A 血清素受体化学探针组

Anat Levit Kaplan, Ryan T Strachan, Joao M Braz, Veronica Craik, Samuel Slocum, Thomas Mangano, Vanessa Amabo, Henry O'Donnell, Parnian Lak, Allan I Basbaum, Bryan L Roth, Brian K Shoichet

Discovery of Human Signaling Systems: Pairing Peptides to G Protein-Coupled Receptors

发现人类信号系统:肽与 G 蛋白偶联受体的配对

Simon R Foster, Alexander S Hauser, Line Vedel, Ryan T Strachan, Xi-Ping Huang, Ariana C Gavin, Sushrut D Shah, Ajay P Nayak, Linda M Haugaard-Kedström, Raymond B Penn, Bryan L Roth, Hans Bräuner-Osborne, David E Gloriam

VEGAS as a Platform for Facile Directed Evolution in Mammalian Cells

VEGAS作为哺乳动物细胞中简易定向进化的平台

Justin G English,Reid H J Olsen,Katherine Lansu,Michael Patel,Karoline White,Adam S Cockrell,Darshan Singh,Ryan T Strachan,Daniel Wacker,Bryan L Roth

Structure of the Nanobody-Stabilized Active State of the Kappa Opioid Receptor

纳米抗体稳定的 Kappa 阿片受体活性状态的结构

Tao Che, Susruta Majumdar, Saheem A Zaidi, Pauline Ondachi, John D McCorvy, Sheng Wang, Philip D Mosier, Rajendra Uprety, Eyal Vardy, Brian E Krumm, Gye Won Han, Ming-Yue Lee, Els Pardon, Jan Steyaert, Xi-Ping Huang, Ryan T Strachan, Alexandra R Tribo, Gavril W Pasternak, F Ivy Carroll, Raymond C St

Mdm2 regulates cardiac contractility by inhibiting GRK2-mediated desensitization of β-adrenergic receptor signaling

Mdm2 通过抑制 GRK2 介导的 β-肾上腺素受体信号脱敏来调节心脏收缩力

Pierre-Yves Jean-Charles, Samuel Mon-Wei Yu, Dennis Abraham, Reddy Peera Kommaddi, Lan Mao, Ryan T Strachan, Zhu-Shan Zhang, Dawn E Bowles, Leigh Brian, Jonathan A Stiber, Stephen N Jones, Walter J Koch, Howard A Rockman, Sudha K Shenoy

Allosteric "beta-blocker" isolated from a DNA-encoded small molecule library

从 DNA 编码的小分子库中分离出的变构“β受体阻滞剂”

Seungkirl Ahn, Alem W Kahsai, Biswaranjan Pani, Qin-Ting Wang, Shuai Zhao, Alissa L Wall, Ryan T Strachan, Dean P Staus, Laura M Wingler, Lillian D Sun, Justine Sinnaeve, Minjung Choi, Ted Cho, Thomas T Xu, Gwenn M Hansen, Michael B Burnett, Jane E Lamerdin, Daniel L Bassoni, Bryant J Gavino, Gitte

Conformationally selective RNA aptamers allosterically modulate the β2-adrenoceptor

构象选择性 RNA 适体变构调节 β2-肾上腺素能受体

Alem W Kahsai, James W Wisler, Jungmin Lee, Seungkirl Ahn, Thomas J Cahill Iii, S Moses Dennison, Dean P Staus, Alex R B Thomsen, Kara M Anasti, Biswaranjan Pani, Laura M Wingler, Hemant Desai, Kristin M Bompiani, Ryan T Strachan, Xiaoxia Qin, S Munir Alam, Bruce A Sullenger, Robert J Lefkowitz1